Synthesis and hybridization property of an oligonucleotide containing a 3-thioformacetal linked pentathymidylate

Bioorg Med Chem Lett. 1999 Feb 8;9(3):319-22. doi: 10.1016/s0960-894x(98)00741-0.

Abstract

A pentathymidylate fully substituted with 3'-thioformacetal intemucleotidic linkages was synthesized and subsequently incorporated into an oligonucleotide (ON) 15mer. Tm analysis was performed on the resulting ON hybridized with its complementary RNA. This duplex demonstrated slightly improved binding affinity relative to the control phosphate diester ON/RNA hybrid.

MeSH terms

  • Acetals / chemistry*
  • Base Sequence
  • Nucleic Acid Hybridization
  • RNA / metabolism
  • Sulfides / chemistry*
  • Thymine Nucleotides / chemical synthesis*
  • Thymine Nucleotides / chemistry
  • Thymine Nucleotides / metabolism

Substances

  • Acetals
  • Sulfides
  • Thymine Nucleotides
  • RNA