Chronic hyperammonemia in rats impairs activation of soluble guanylate cyclase in neurons and in lymphocytes: a putative peripheral marker for neurological alterations

Biochem Biophys Res Commun. 1999 Apr 13;257(2):405-9. doi: 10.1006/bbrc.1999.0486.

Abstract

Chronic hyperammonemia impairs the glutamate-nitric oxide-cGMP pathway in rat brain in vivo. The aims of this work were to assess whether hyperammonemia impairs modulation of soluble guanylate cyclase, and to look for a peripheral marker for impairment of this pathway in brain. We activated the pathway at different steps using glutamate, SNAP, or YC-1. In control neurons these compounds increased cGMP by 7.4-, 9.7- and 7.2-fold, respectively. In ammonia-treated neurons formation of cGMP induced by glutamate, SNAP, and YC-1 was reduced by 50%, 56%, and 52%, respectively, indicating that hyperammonemia impairs activation of guanylate cyclase. This enzyme is also present in lymphocytes. Activation of guanylate cyclase by SNAP or YC-1 was impaired in lymphocytes from hyperammonemic rats. These results suggest that determination of the activation of soluble guanylate cyclase in lymphocytes could serve as a peripheral marker for impairment of the neuronal glutamate-nitric oxide-cGMP pathway in brain.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Ammonia / metabolism
  • Ammonia / pharmacology*
  • Animals
  • Biomarkers / analysis
  • Cells, Cultured
  • Chronic Disease
  • Cyclic GMP / metabolism
  • Enzyme Activation / drug effects
  • Excitatory Amino Acid Antagonists / pharmacology
  • Glutamic Acid / pharmacology
  • Guanylate Cyclase / biosynthesis*
  • Hepatic Encephalopathy / etiology
  • Hepatic Encephalopathy / metabolism*
  • Hepatic Encephalopathy / pathology
  • Indazoles / antagonists & inhibitors
  • Indazoles / pharmacology
  • Lymphocytes / drug effects
  • Lymphocytes / enzymology*
  • Lymphocytes / metabolism
  • Neurons / drug effects
  • Neurons / enzymology*
  • Neurons / metabolism
  • Penicillamine / analogs & derivatives
  • Penicillamine / antagonists & inhibitors
  • Penicillamine / pharmacology
  • Rats
  • Rats, Wistar
  • S-Nitroso-N-Acetylpenicillamine
  • Time Factors

Substances

  • Biomarkers
  • Excitatory Amino Acid Antagonists
  • Indazoles
  • 3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazole
  • Glutamic Acid
  • Ammonia
  • S-Nitroso-N-Acetylpenicillamine
  • Guanylate Cyclase
  • Penicillamine
  • Cyclic GMP