Neuregulin-4: a novel growth factor that acts through the ErbB-4 receptor tyrosine kinase

Oncogene. 1999 Apr 29;18(17):2681-9. doi: 10.1038/sj.onc.1202631.

Abstract

The ErbB/HER family of receptor tyrosine kinases consists of four receptors that bind a large number of growth factor ligands sharing an epidermal growth factor- (EGF)-like motif. Whereas ErbB-1 binds seven different ligands whose prototype is EGF, the three families of neuregulins (NRGs) activate ErbB-3 and/or ErbB-4. Here we characterize a fourth neuregulin, NRG-4, that acts through ErbB-4. The predicted pro-NRG-4 is a transmembrane protein carrying a unique EGF-like motif and a short cytoplasmic domain. A synthetic peptide encompassing the full-length EGF-like domain can induce growth of interleukin-dependent cells ectopically expressing ErbB-4, but not cells expressing the other three ErbB proteins or their combinations. Consistent with specificity to ErbB-4, NRG-4 can displace an ErbB-4-bound NRG-1 and can activate signaling downstream of this receptor. Expression of NRG-4 mRNA was detected in the adult pancreas and weakly in muscle; other tissues displayed no detectable NRG-4 mRNA. The primary structure and the pattern of expression of NRG-4, together with the strict specificity of this growth factor to ErbB-4, suggest a physiological role distinct from that of the known ErbB ligands.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Base Sequence
  • Cell Division / physiology
  • ErbB Receptors / physiology*
  • Glycoproteins / physiology*
  • Humans
  • Ligands
  • Molecular Sequence Data
  • Nerve Growth Factors / physiology*
  • Neuregulins
  • Organ Specificity
  • Protein Structure, Tertiary
  • RNA, Messenger / biosynthesis
  • Receptor, ErbB-4

Substances

  • Glycoproteins
  • Ligands
  • Nerve Growth Factors
  • Neuregulins
  • RNA, Messenger
  • ERBB4 protein, human
  • ErbB Receptors
  • Receptor, ErbB-4

Associated data

  • GENBANK/AF083067