A fusion protein of interleukin-11 and soluble interleukin-11 receptor acts as a superagonist on cells expressing gp130

FEBS Lett. 1999 Apr 30;450(1-2):117-22. doi: 10.1016/s0014-5793(99)00477-9.

Abstract

Interleukin-11 is a hematopoietic cytokine that signals via the signal transducer gp130. Although gp130 is ubiquitously expressed, interleukine-11 responsiveness is restricted to cells that express the interleukine-11 receptor alpha-subunit. The interleukine-11 receptor alpha-subunit can be functionally replaced by its soluble form indicating that the transmembrane and cytoplasmic parts are not required for signal transduction. Here, we show that a recombinant fusion protein of a fragment of the human interleukine-11 receptor alpha-subunit ectodomain linked to human interleukine-11 acts as a superagonist on cells expressing gp130 but lacking the membrane-bound interleukine-11 receptor alpha-subunit. It induces acute phase protein synthesis in hepatoma cells and efficiently promotes proliferation of Ba/F3 cells stably, transfected with gp130. In these bioassays, the fusion protein of a fragment of the human interleukine-11 receptor alpha-subunit ectodomain linked to human interleukine-11 is 50 times more potent than the combination of interleukine-11 and the soluble interleukine-11 receptor alpha-subunit. Thus, our findings support the concept that covalent fusion of two soluble proteins required for receptor activation dramatically increases their bioactivity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute-Phase Proteins / biosynthesis
  • Amino Acid Sequence
  • Antigens, CD / metabolism*
  • Antigens, CD / pharmacology
  • Cytokine Receptor gp130
  • DNA-Binding Proteins / metabolism
  • Gene Expression
  • Humans
  • Interleukin-11 / genetics*
  • Interleukin-11 / metabolism
  • Interleukin-11 Receptor alpha Subunit
  • Membrane Glycoproteins / metabolism*
  • Membrane Glycoproteins / pharmacology
  • Molecular Sequence Data
  • Pichia / genetics
  • Protease Inhibitors / metabolism
  • Receptors, Interleukin / genetics*
  • Receptors, Interleukin / metabolism
  • Receptors, Interleukin-11
  • Recombinant Fusion Proteins / metabolism*
  • STAT1 Transcription Factor
  • STAT3 Transcription Factor
  • Trans-Activators / metabolism
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Acute-Phase Proteins
  • Antigens, CD
  • DNA-Binding Proteins
  • IL11RA protein, human
  • IL6ST protein, human
  • Interleukin-11
  • Interleukin-11 Receptor alpha Subunit
  • Membrane Glycoproteins
  • Protease Inhibitors
  • Receptors, Interleukin
  • Receptors, Interleukin-11
  • Recombinant Fusion Proteins
  • STAT1 Transcription Factor
  • STAT1 protein, human
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • Trans-Activators
  • Cytokine Receptor gp130