A direct comparison of the activities of two humanized respiratory syncytial virus monoclonal antibodies: MEDI-493 and RSHZl9

J Infect Dis. 1999 Jul;180(1):35-40. doi: 10.1086/314846.

Abstract

Two humanized monoclonal antibodies, MEDI-493 and RSHZ19, were developed independently as potential improvements over RSV-IGIV for prevention of respiratory syncytial virus (RSV) infection. RSV-IGIV is a polyclonal human antibody preparation for intravenous infusion enriched for RSV neutralizing activity. A phase III clinical trial showed that MEDI-493 significantly reduced hospitalizations due to RSV infection. In a separate trial, RSHZ19 failed to show significant efficacy. In new studies, the in vitro and in vivo activities of MEDI-493 and RSHZ19 were compared to determine whether the different clinical results are related to differences in biologic activity. MEDI-493 was consistently 4- to 5-fold more potent than RSHZ19 in antigen binding, RSV neutralization, and fusion inhibition assays. Although both MEDI-493 and RSHZ19 were effective against A and B subtypes of RSV in the cotton rat model of RSV infection, 2- to 4-fold higher doses of RSHZ19 were required for similar protection. The enhanced activity of MEDI-493 compared with RSHZ19 may, in part, explain its better clinical effect.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Antibodies, Monoclonal / immunology*
  • Antibodies, Monoclonal / therapeutic use
  • Antibodies, Monoclonal, Humanized
  • Antibody Affinity
  • Cell Fusion / drug effects
  • Dose-Response Relationship, Drug
  • HN Protein*
  • Immunoglobulin G / immunology
  • Immunotherapy
  • Neutralization Tests
  • Palivizumab
  • Respiratory Syncytial Virus Infections / drug therapy*
  • Respiratory Syncytial Viruses / immunology*
  • Sigmodontinae
  • Viral Envelope Proteins
  • Viral Fusion Proteins / immunology
  • Viral Proteins / immunology

Substances

  • Antibodies, Monoclonal
  • Antibodies, Monoclonal, Humanized
  • HN Protein
  • Immunoglobulin G
  • RSHZ19 monoclonal antibody
  • Viral Envelope Proteins
  • Viral Fusion Proteins
  • Viral Proteins
  • attachment protein G
  • Palivizumab