A TSH/dibutyryl cAMP activated Cl-/I- channel in FRTL-5 cells

Biochem Biophys Res Commun. 1999 Jun 16;259(3):631-5. doi: 10.1006/bbrc.1999.0836.

Abstract

An iodide (I) and chloride (Cl) channel has been identified in the continuously cultured FRTL-5 thyroid cell line using a cell attached patch clamp technique. The channel is activated by TSH and dibutyryladenosine cyclic monophosphate (Bt2-cAMP) but not by phorbol 12-myristate 13-acetate (TPA). Gluconate can not replace chloride or iodide and the channel is impermeable to Na+,K+ and tetraethylammonium ions. The current-voltage relationship demonstrates that the single channel current is a linear function of the clamp voltage. Single channel currents reversed at a pipette potential close to 0 mV. The mean single channel conductance was 60 pS for Cl- and 50 pS for I-. From the I-V relationship there was a strong outward rectification with Cl-, and a complete block with I-, in the single channel current above +40 mV. The feature of the channel is manifested in the single channel records by four distinct, equally spaced conductance levels. We suggest the channel is important for the transport of I and Cl ions across the apical membrane into the colloid space and is important for hormone synthesis and follicle formation.

MeSH terms

  • Animals
  • Bucladesine / pharmacology*
  • Calcium Channels / physiology*
  • Cells, Cultured
  • Iodine / physiology*
  • Ion Channels / physiology*
  • Patch-Clamp Techniques
  • Rats
  • Tetradecanoylphorbol Acetate / metabolism
  • Thyroid Gland / metabolism
  • Thyrotropin / metabolism*

Substances

  • Calcium Channels
  • Ion Channels
  • Bucladesine
  • Thyrotropin
  • Iodine
  • Tetradecanoylphorbol Acetate