Synthesis and antibacterial activity of 2-aryl-2,5-dihydro-3(3H)-oxo-pyridazino[4,3-b]indole-4-carboxylic acids

Farmaco. 1999 Mar 31;54(3):191-4. doi: 10.1016/s0014-827x(99)00021-x.

Abstract

The in vitro antibacterial and antifungal activities of a series of pyridazinoindolonic acids II against some selected representative of Gram-positive, Gram-negative bacteria and fungi have been investigated. Some interesting observations among the structural features necessary for high antibacterial activity are presented and discussed.

MeSH terms

  • Anti-Bacterial Agents / chemical synthesis
  • Anti-Bacterial Agents / pharmacology*
  • Indoles / chemical synthesis
  • Indoles / pharmacology*
  • Molecular Structure
  • Pyridazines / chemical synthesis
  • Pyridazines / pharmacology*

Substances

  • Anti-Bacterial Agents
  • Indoles
  • Pyridazines