Abstract
In an aortic smooth muscle cell line, A10 cells, we investigated the effect of sphingosine 1-phosphate on the induction of heat shock protein 27 (HSP27), a low-molecular-weight heat shock protein. Sphingosine 1-phosphate significantly induced the accumulation of HSP27 in a pertussis toxin-sensitive manner. The effect was dose-dependent in the range between 0.1 and 30 microM. Sphingosine 1-phosphate stimulated an increase in the levels of mRNA for HSP27. Sphingosine 1-phosphate stimulated both p42/p44 mitogen-activated protein (MAP) kinase and p38 MAP kinase activation. PD98059, an inhibitor of the upstream kinase that activates p42/p44 MAP kinase, did not affect sphingosine 1-phosphate-stimulated HSP27 induction. In contrast, SB203580, an inhibitor of p38 MAP kinase, reduced sphingosine 1-phosphate-induced HSP27 induction. SB203580 reduced the levels of mRNA for HSP27 induced by sphingosine 1-phosphate. These results indicate that sphingosine 1-phosphate stimulates the induction of HSP27 via p38 MAP kinase activation in aortic smooth muscle cells.
Copyright 1999 Academic Press.
MeSH terms
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Animals
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Aorta
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Calcium-Calmodulin-Dependent Protein Kinases / antagonists & inhibitors
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Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
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Cell Line
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Dose-Response Relationship, Drug
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Enzyme Activation / drug effects
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Flavonoids / pharmacology
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Gene Expression Regulation / drug effects
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Heat-Shock Proteins / biosynthesis*
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Heat-Shock Proteins / genetics
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Imidazoles / pharmacology
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Lysophospholipids*
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Mitogen-Activated Protein Kinase 1 / antagonists & inhibitors
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Mitogen-Activated Protein Kinase 1 / metabolism
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Mitogen-Activated Protein Kinase 3
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Mitogen-Activated Protein Kinases*
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Muscle, Smooth, Vascular / cytology
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Muscle, Smooth, Vascular / drug effects
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Muscle, Smooth, Vascular / enzymology
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Muscle, Smooth, Vascular / metabolism*
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Pertussis Toxin
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Phosphorylation / drug effects
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Pyridines / pharmacology
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RNA, Messenger / genetics
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RNA, Messenger / metabolism
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Rats
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Signal Transduction / drug effects*
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Sphingosine / analogs & derivatives*
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Sphingosine / antagonists & inhibitors
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Sphingosine / pharmacology
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Virulence Factors, Bordetella / pharmacology
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p38 Mitogen-Activated Protein Kinases
Substances
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Flavonoids
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Heat-Shock Proteins
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Imidazoles
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Lysophospholipids
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Pyridines
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RNA, Messenger
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Virulence Factors, Bordetella
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sphingosine 1-phosphate
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Pertussis Toxin
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Calcium-Calmodulin-Dependent Protein Kinases
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Mitogen-Activated Protein Kinase 1
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Mitogen-Activated Protein Kinase 3
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Mitogen-Activated Protein Kinases
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p38 Mitogen-Activated Protein Kinases
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Sphingosine
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SB 203580
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2-(2-amino-3-methoxyphenyl)-4H-1-benzopyran-4-one