Mutated N-ras upregulates Bcl-2 in human melanoma in vitro and in SCID mice

Melanoma Res. 1999 Aug;9(4):347-50. doi: 10.1097/00008390-199908000-00002.

Abstract

Activation of the N-ras gene by point mutation occurs in about 15% of all human melanomas. In recently established severe combined immunodeficiency (SCID) mouse xenotransplantation models for human melanoma, we demonstrated that mutated N-ras not only contributes to tumour growth by enhancing cellular proliferation, but also by blocking apoptosis. Mutated N-ras overexpression protected human melanomas from naturally occurring apoptosis and, in a more pronounced way, from chemotherapy-induced apoptosis in vitro and in vivo. Given the potential clinical importance of these findings we sought to determine the underlying mechanism. We found that mutated N-ras specifically upregulates the expression of the anti-apoptosis gene bcl-2 in two human melanoma cell lines in vitro and in SCID mice. Neither the expression of the anti-apoptotic protein Bcl-xL nor that of the pro-apoptotic proteins Bax and Bak were altered in cells expressing mutated N-Ras. The increase in Bcl-2 expression mediated by mutated ras therefore qualifies as a rational explanation for the enhanced chemoresistance of human melanoma expressing mutated N-Ras.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis
  • Blotting, Western
  • Gene Expression Regulation, Neoplastic*
  • Genes, ras / genetics*
  • Humans
  • Melanoma / genetics*
  • Melanoma / metabolism*
  • Melanoma / pathology
  • Membrane Proteins / biosynthesis
  • Mice
  • Mice, SCID
  • Neoplasm Transplantation
  • Point Mutation
  • Proto-Oncogene Proteins / biosynthesis
  • Proto-Oncogene Proteins c-bcl-2 / biosynthesis*
  • Transfection
  • Tumor Cells, Cultured
  • Up-Regulation / genetics*
  • bcl-2 Homologous Antagonist-Killer Protein
  • bcl-2-Associated X Protein
  • bcl-X Protein

Substances

  • BAK1 protein, human
  • BAX protein, human
  • BCL2L1 protein, human
  • Bak1 protein, mouse
  • Bax protein, mouse
  • Bcl2l1 protein, mouse
  • Membrane Proteins
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-bcl-2
  • bcl-2 Homologous Antagonist-Killer Protein
  • bcl-2-Associated X Protein
  • bcl-X Protein