Ligand-induced ubiquitination of the epidermal growth factor receptor involves the interaction of the c-Cbl RING finger and UbcH7

J Biol Chem. 1999 Oct 29;274(44):31707-12. doi: 10.1074/jbc.274.44.31707.

Abstract

c-Cbl plays a negative regulatory role in tyrosine kinase signaling by an as yet undefined mechanism. We demonstrate here, using the yeast two-hybrid system and an in vitro binding assay, that the c-Cbl RING finger domain interacts with UbcH7, a ubiquitin-conjugating enzyme (E2). UbcH7 interacted with the wild-type c-Cbl RING finger domain but not with a RING finger domain that lacks the amino acids that are deleted in 70Z-Cbl, an oncogenic mutant of c-Cbl. The in vitro interaction was enhanced by sequences on both the N- and C-terminal sides of the RING finger. In vivo and in vitro experiments revealed that c-Cbl and UbcH7 synergistically promote the ligand-induced ubiquitination of the epidermal growth factor receptor (EGFR). In contrast, 70Z-Cbl markedly reduced the ligand-induced, UbcH7-mediated ubiquitination of the EGFR. MG132, a proteasome inhibitor, significantly prolonged the ligand-induced phosphorylation of both the EGFR and c-Cbl. Thus, c-Cbl plays an essential role in the ligand-induced ubiquitination of the EGFR by a mechanism that involves an interaction of the RING finger domain with UbcH7. This mechanism participates in the down-regulation of tyrosine kinase receptors and loss of this function, as occurs in the naturally occurring 70Z-Cbl isoform, probably contributes to oncogenic transformation.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Cysteine Endopeptidases / drug effects
  • Cysteine Endopeptidases / metabolism
  • Cysteine Proteinase Inhibitors / pharmacology
  • Epidermal Growth Factor / metabolism*
  • ErbB Receptors / metabolism*
  • Leupeptins / pharmacology
  • Ligands
  • Ligases / metabolism*
  • Models, Biological
  • Multienzyme Complexes / drug effects
  • Multienzyme Complexes / metabolism
  • Phosphorylation
  • Proteasome Endopeptidase Complex
  • Protein Binding
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-cbl
  • Recombinant Fusion Proteins / metabolism
  • Two-Hybrid System Techniques
  • Tyrosine / metabolism
  • Ubiquitin-Conjugating Enzymes*
  • Ubiquitin-Protein Ligases*
  • Ubiquitins / metabolism*
  • Zinc Fingers

Substances

  • Cysteine Proteinase Inhibitors
  • Leupeptins
  • Ligands
  • Multienzyme Complexes
  • Proto-Oncogene Proteins
  • Recombinant Fusion Proteins
  • Ubiquitins
  • Tyrosine
  • Epidermal Growth Factor
  • UBE2L3 protein, human
  • Ubiquitin-Conjugating Enzymes
  • Proto-Oncogene Proteins c-cbl
  • Ubiquitin-Protein Ligases
  • ErbB Receptors
  • Cysteine Endopeptidases
  • Proteasome Endopeptidase Complex
  • Ligases
  • CBL protein, human
  • benzyloxycarbonylleucyl-leucyl-leucine aldehyde