Kinetics and inhibition of cyclomaltodextrinase from alkalophilic Bacillus sp. I-5

Arch Biochem Biophys. 2000 Jan 1;373(1):110-5. doi: 10.1006/abbi.1999.1471.

Abstract

The cyclomaltodextrinase from alkalophilic Bacillus sp. I-5 (CDase I-5) was expressed in Escherichia coli and the purified enzyme was used for characterization of the enzyme action. The hydrolysis products were monitored by both HPLC and high-performance ion chromatography analysis that enable the kinetic analysis of the cyclomaltodextrin (CD)-degrading reaction. Analysis of the kinetics of cyclomaltodextrin hydrolysis by CDase I-5 indicated that ring-opening of the cyclomaltodextrin was the major limiting step and that CDase I-5 preferentially degraded the linear maltodextrin chain by removing the maltose unit. The substrate binding affinity of the enzyme was almost same for those of cyclomaltodextrins while the rate of ring-opening was the fastest for cyclomaltoheptaose. Acarbose and methyl 6-amino-6-deoxy-alpha-d-glucopyranoside were relatively strong competitive inhibitors with K(i) values of 1.24 x 10(-3) and 8.44 x 10(-1) mM, respectively. Both inhibitors are likely to inhibit the ring-opening step of the CD degradation reaction.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acarbose / pharmacology
  • Bacillus / enzymology*
  • Bacillus / genetics
  • Cyclodextrins / metabolism
  • Escherichia coli / genetics
  • Glucosides / pharmacology
  • Glycoside Hydrolases / antagonists & inhibitors*
  • Glycoside Hydrolases / genetics
  • Glycoside Hydrolases / metabolism*
  • Kinetics
  • Recombinant Proteins / antagonists & inhibitors
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism
  • Substrate Specificity

Substances

  • Cyclodextrins
  • Glucosides
  • Recombinant Proteins
  • methyl-6-amino-6-deoxyglucopyranoside
  • Glycoside Hydrolases
  • cyclomaltodextrinase
  • Acarbose