Ivermectin: concentration-dependent effects on adenosine triphosphatases in adult worms of Onchocerca volvulus

Acta Trop. 2000 Jan 5;74(1):7-11. doi: 10.1016/s0001-706x(99)00052-2.

Abstract

The effect of increasing concentrations of ivermectin on adenosine triphosphatase (ATPase) activity was investigated in adult worms of Onchocerca volvulus. Mean Mg- and Na,K-ATPase activities decreased significantly (F ratio = 29.82, P < 0.01 and F ratio = 28.54, P < 0.01, respectively) with increasing concentrations of ivermectin (0-100 ng/ml) in the female worms. When male and female worms were mixed with equal amounts of proteins from each, only the Na,K-ATPase activity was significantly decreased (F ratio = 56.61, P < 0.01) over a similar range of ivermectin concentrations. Since ivermectin exhibits concentration-dependent effects on both ATPases in female adult worms, this might provide an insight into other effects of the drug. However, the adjustment of the dose of ivermectin to obtain a nodular concentration of at least 40 ng/ml is therefore recommended in the complete chemotherapy of onchocerciasis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphatases / drug effects*
  • Adenosine Triphosphatases / metabolism
  • Adult
  • Analysis of Variance
  • Animals
  • Antiprotozoal Agents / pharmacology*
  • Dose-Response Relationship, Drug
  • Female
  • Humans
  • Ivermectin / pharmacology*
  • Male
  • Nigeria
  • Onchocerca volvulus / drug effects*
  • Onchocerca volvulus / enzymology

Substances

  • Antiprotozoal Agents
  • Ivermectin
  • Adenosine Triphosphatases