Conversion from thrice daily to twice daily administration of gabapentin (GBP) in partial epilepsy: analysis of clinical efficacy and plasma levels

Seizure. 2000 Jan;9(1):47-50. doi: 10.1053/seiz.1999.0340.

Abstract

Gabapentin has been administered in placebo-controlled studies with a thrice daily (T.I.D.) schedule, because of its short half-life. However, clinical efficacy does not seem strictly related to plasma levels: a twice daily (B.I.D.) schedule might therefore be possible. The aim of our study was to verify if the conversion from a T.I.D. to a B.I.D. regimen affected the efficacy and safety of gabapentin therapy. Out of 171 patients treated with add-on gabapentin, we selected 29 stable responders, who were followed for three months with a T.I.D. schedule and then switched to B.I.D. regimen for further three months. Seizure number, side-effects and trough plasma levels of gabapentin were collected during both periods. Gabapentin mean dose was 2117.2 mg/day. Mean number of seizures/months was: 4.2 at baseline, 1.0 during the T.I.D., and 0.9 during the B.I.D. period. Mean trough plasma level of gabapentin was 5.9 microgram/ml during the T.I.D. and 5.2 microgram/ml during the B.I.D. period. Twelve side-effects were reported by 11 patients during the T.I.D. and 6 by 5 patients during the B.I.D. period., sedation and vertigo were the most frequent in both. Results of our study suggest that gabapentin can be administered safely and effectively either with a T.I.D. and a B.I.D. regimen.

Publication types

  • Clinical Trial

MeSH terms

  • Acetates / administration & dosage*
  • Acetates / blood*
  • Acetates / pharmacokinetics
  • Adolescent
  • Adult
  • Amines*
  • Anticonvulsants / administration & dosage*
  • Anticonvulsants / blood*
  • Anticonvulsants / pharmacokinetics
  • Cross-Over Studies
  • Cyclohexanecarboxylic Acids*
  • Drug Administration Schedule
  • Epilepsies, Partial / drug therapy*
  • Female
  • Gabapentin
  • Humans
  • Male
  • Middle Aged
  • Polypharmacy
  • Treatment Outcome
  • gamma-Aminobutyric Acid*

Substances

  • Acetates
  • Amines
  • Anticonvulsants
  • Cyclohexanecarboxylic Acids
  • gamma-Aminobutyric Acid
  • Gabapentin