Improvement in left ventricular function in response to carvedilol is accompanied by attenuation of neurohumoral activation in patients with dilated cardiomyopathy

J Card Fail. 2000 Mar;6(1):3-10. doi: 10.1016/s1071-9164(00)80004-4.

Abstract

Background: We sought to evaluate whether improvement in ejection fraction (EF) with carvedilol therapy is accompanied by improvement in neurohumoral factors.

Methods and results: Forty-two patients with dilated cardiomyopathy were given carvedilol for 3 to 5 months. Changes in EF, plasma atrial natriuretic peptide (ANP), brain natriuretic peptide (BNP), and norepinephrine levels were determined. Iodine-123 metaiodobenzylguanidine (MIBG) images were also obtained before and after carvedilol therapy. Myocardial uptake of MIBG was calculated as the heart to mediastinal activity ratio (H/M). Storage and release of MIBG was calculated as percent myocardial MIBG washout rate (WR). We divided patients into 2 groups: 27 responders whose EF increased by more than 5% and 15 nonresponders whose EF increased by 5% or less. EF of responders increased by 15 +/- 5% and that of nonresponders by 1 +/- 4%. Although MIBG image-derived indexes of nonresponders remained unchanged, the delayed H/M (1.91 +/- 0.34 v 2.24 +/- 0.53, P < .01) and WR (49 +/- 11 v 39 +/- 9%, P < .01) of responders improved, respectively. The plasma ANP (51 +/- 50 v 27 +/- 24 pg/mL, P < .01) and BNP (194 +/- 197 v 49 +/- 62 pg/mL, P < .01) levels of responders decreased. The degree of changes in the plasma BNP level correlated with changes in EF (r = -.698, P < .01).

Conclusion: The improvement in EF with carvedilol therapy was proved to be accompanied by an improvement in neurohumoral factors.

Publication types

  • Comparative Study

MeSH terms

  • 3-Iodobenzylguanidine
  • Adrenergic beta-Antagonists / therapeutic use*
  • Adult
  • Aged
  • Atrial Natriuretic Factor / blood*
  • Biomarkers / blood
  • Carbazoles / therapeutic use*
  • Cardiomyopathy, Dilated / blood
  • Cardiomyopathy, Dilated / drug therapy*
  • Cardiomyopathy, Dilated / physiopathology
  • Carvedilol
  • Female
  • Heart Ventricles / diagnostic imaging
  • Heart Ventricles / drug effects
  • Heart Ventricles / physiopathology
  • Humans
  • Male
  • Middle Aged
  • Natriuretic Peptide, Brain / blood*
  • Norepinephrine / blood*
  • Propanolamines / therapeutic use*
  • Radiopharmaceuticals
  • Recovery of Function
  • Retrospective Studies
  • Stroke Volume / drug effects
  • Tomography, Emission-Computed, Single-Photon
  • Treatment Outcome
  • Ventricular Function, Left / drug effects
  • Ventricular Function, Left / physiology*

Substances

  • Adrenergic beta-Antagonists
  • Biomarkers
  • Carbazoles
  • Propanolamines
  • Radiopharmaceuticals
  • Carvedilol
  • Natriuretic Peptide, Brain
  • 3-Iodobenzylguanidine
  • Atrial Natriuretic Factor
  • Norepinephrine