Disulfide bond formation is not required for human chorionic gonadotropin subunit association. Studies with dithiothreitol in JEG-3 cells

J Biol Chem. 2000 Apr 21;275(16):11765-70. doi: 10.1074/jbc.275.16.11765.

Abstract

To study the influence of disulfide bridge formation on the assembly of the subunits of human chorionic gonadotropin in JEG-3 choriocarcinoma cells, dithiothreitol (DTT) was used to create a reducing milieu in the endoplasmic reticulum (ER) in vivo. In the presence of 5 mM DTT during pulse-chase experiments all of the beta-subunit precursors observed in unperturbed cells (pbeta(0), pbeta(1), pbeta(2), and beta(*)) collapsed into the pbeta(0) form. The reducing milieu of the ER was reoxidized in less than 5 min after removal of DTT from the medium. DTT markedly increased the half-life of the pbeta(0) precursor from 8.8 to 65.2 min. Under reoxidation conditions, the beta-subunit precursors folded back from pbeta(0) in less than 5 min. In unperturbed JEG-3 cells, the alpha-subunit was present in both fully glycosylated and monoglycosylated precursor (pre-alpha) forms. The attachment of the second N-linked glycan residue of the alpha-subunit was accelerated in the presence of DTT, and consequently pre-alpha-subunit was missing from the DTT-treated cultures. The formation of alphabeta-dimers appeared to be at least partially independent of the oxidation state in the ER. The alphabeta-dimer was present under conditions in which disulfide bridge formation was prevented by exposure to 5 mM DTT before and during the pulse period. This clearly suggests that the human chorionic gonadotropin subunits may acquire association-competent conformations even when no disulfide bridge formation has taken place.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Chorionic Gonadotropin, beta Subunit, Human / chemistry
  • Chorionic Gonadotropin, beta Subunit, Human / metabolism*
  • Disulfides / metabolism*
  • Dithiothreitol / metabolism*
  • Electrophoresis, Polyacrylamide Gel
  • Glycoprotein Hormones, alpha Subunit / chemistry
  • Glycoprotein Hormones, alpha Subunit / metabolism*
  • Glycosylation
  • Humans
  • Kinetics
  • Protein Conformation
  • Tumor Cells, Cultured

Substances

  • Chorionic Gonadotropin, beta Subunit, Human
  • Disulfides
  • Glycoprotein Hormones, alpha Subunit
  • Dithiothreitol