Analgesic principle from Abutilon indicum

Pharmazie. 2000 Apr;55(4):314-6.

Abstract

Bioactivity guided isolation of Abutilon indicum yielded eugenol [4-allyl-2-methoxyphenol], which was found to possess significant analgesic activity. At doses of 10, 30, and 50 mg/kg body weight, eugenol exhibited 21.30 (p < 0.05), 42.25 (p < 0.01) and 92.96% (p < 0.001) inhibition of acetic acid induced writhing in mice. At a dose of 50 mg/kg body weight, eugenol showed 33.40% (p < 0.05) prolongation of tail flicking time determined by the radiant heat method.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetates
  • Analgesics / isolation & purification
  • Analgesics / pharmacology*
  • Animals
  • Chromatography, Thin Layer
  • Eugenol / analogs & derivatives*
  • Eugenol / isolation & purification
  • Eugenol / pharmacology
  • Hot Temperature
  • Male
  • Mice
  • Oils, Volatile / chemistry
  • Pain Measurement / drug effects
  • Plants, Medicinal / chemistry*
  • Rats

Substances

  • Acetates
  • Analgesics
  • Oils, Volatile
  • eugenol-4-allyl-2-methoxyphenol
  • Eugenol