Preparation and characterization of solid lipid nanospheres containing paclitaxel

Eur J Pharm Sci. 2000;10(4):305-9. doi: 10.1016/s0928-0987(00)00081-6.

Abstract

The study describes the development of stealth and non-stealth solid lipid nanospheres (SLNs) as colloidal carriers for paclitaxel, a drug with very low solubility. SLNs are constituted mainly of bioacceptable and biodegradable lipids, such as tripalmitin and phosphatidylcholine, and can incorporate amounts of paclitaxel up to 2.8%. Stealth and non-stealth loaded SLNs are in the nanometer size range and can be sterilized and freeze-dried. Thermal analysis (differential scanning calorimetry) showed that paclitaxel is not able to crystallize in the SLNs. Release of paclitaxel from SLNs is very low. Non-stealth and stealth SLNs are stable over time without precipitation of paclitaxel and can be proposed for its parenteral administration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents, Phytogenic / chemistry*
  • Chemistry, Pharmaceutical
  • Drug Carriers
  • Half-Life
  • Paclitaxel / chemistry*
  • Phosphatidylcholines / chemical synthesis*
  • Triglycerides / chemical synthesis*

Substances

  • Antineoplastic Agents, Phytogenic
  • Drug Carriers
  • Phosphatidylcholines
  • Triglycerides
  • tripalmitin
  • Paclitaxel