Thymidine kinase gene therapy with concomitant topotecan chemotherapy for recurrent ovarian cancer

Cancer Gene Ther. 2000 Jun;7(6):839-44. doi: 10.1038/sj.cgt.7700192.

Abstract

Introduction: Patients with recurrent ovarian cancer were treated with a replication-deficient recombinant adenovirus containing the herpes simplex virus thymidine kinase gene administered intraperitoneally (i.p.) followed by administration of an anti-herpetic prodrug and topotecan.

Materials and methods: A total of 10 patients with stage IIIc epithelial ovarian cancer underwent secondary debulking to < or =0.5 cm residual tumor. Patients with normal i.p. flow received i.p. delivery of adenovirus. Two patients each were treated on dose level 1 (2 x 10(10) vector particles (VP)), dose level 2 (2 x 10(11) VP), and dose level 3 (2 x 10(12) VP); four patients were treated on dose level 4 (2 x 10(13) VP). Acyclovir and topotecan were started 24 hours after vector delivery.

Results: No patient treated at any dose level incurred unanticipated toxic effects, and all side effects resolved. The most common adverse event was myelosuppression: grade 3 or 4 thrombocytopenia with grade 2-4 anemia in three patients and grade 3 or 4 neutropenia in eight patients. Three patients developed thrombocytosis and three patients had a mild elevation of serum glutamic pyruvic transaminase/alanine aminotransferase. Temperature elevations that were not associated with detectable infection occurred in two patients.

Discussion: I.p. delivery of adenoviral vector with concomitant topotecan chemotherapy was well tolerated without significant lasting toxicities. Side effects were independent of the dose of adenoviral vector.

Publication types

  • Clinical Trial
  • Clinical Trial, Phase I
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acyclovir / administration & dosage
  • Acyclovir / therapeutic use
  • Adenocarcinoma / therapy
  • Adenocarcinoma, Clear Cell / therapy
  • Adenoviridae / genetics
  • Adult
  • Aged
  • Antiviral Agents / administration & dosage
  • Antiviral Agents / therapeutic use
  • Combined Modality Therapy
  • Cystadenocarcinoma, Papillary / therapy
  • DNA / analysis
  • Enzyme Inhibitors / administration & dosage
  • Enzyme Inhibitors / therapeutic use*
  • Female
  • Follow-Up Studies
  • Gene Transfer Techniques
  • Genetic Therapy / methods*
  • Genetic Vectors
  • Humans
  • Injections, Intraperitoneal
  • Middle Aged
  • Neoplasm Recurrence, Local / therapy*
  • Ovarian Neoplasms / therapy*
  • Polymerase Chain Reaction
  • Thymidine Kinase / genetics*
  • Topotecan / administration & dosage
  • Topotecan / therapeutic use*

Substances

  • Antiviral Agents
  • Enzyme Inhibitors
  • Topotecan
  • DNA
  • Thymidine Kinase
  • Acyclovir