Synthesis and biological properties of new glycosidic cationic lipids for DNA delivery

Bioorg Med Chem Lett. 2000 Jun 19;10(12):1393-5. doi: 10.1016/s0960-894x(00)00251-1.

Abstract

Lipidic glycosides with amino alkyl pendent groups were synthesized and evaluated for in vitro DNA transfection activity. The first representative of this new class of cationic lipids showed good gene delivery and low toxicity to HeLa and 3T3 cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3 Cells
  • Animals
  • Anions
  • DNA / administration & dosage*
  • Glycosides / chemistry*
  • HeLa Cells
  • Humans
  • Lipids / chemical synthesis*
  • Lipids / chemistry
  • Lipids / pharmacology*
  • Mice

Substances

  • Anions
  • Glycosides
  • Lipids
  • DNA