Osteoprotegerin ligand modulates murine osteoclast survival in vitro and in vivo

Am J Pathol. 2000 Aug;157(2):435-48. doi: 10.1016/S0002-9440(10)64556-7.

Abstract

Osteoprotegerin ligand (OPGL) targets osteoclast precursors and osteoclasts to enhance differentiation and activation, however, little is known about OPGL effects on osteoclast survival. In vitro, the combination of OPGL + colony-stimulating factor-1 (CSF-1) is required for optimal osteoclast survival. Ultrastructurally, apoptotic changes were observed in detached cells and culture lysates exhibited elevated caspase 3 activity, particularly in cultures lacking CSF-1. DEVD-FMK (caspase 3 inhibitor) partially protected cells when combined with OPGL, but not when used alone or in combination with CSF-1. CSF-1 maintained NF-kappaB activation and increased the expression of bcl-2 and bcl-X(L) mRNA, but had no effect on JNK activation. In contrast, OPGL enhanced both NF-kappaB and JNK kinase activation and increased the expression of c-src, but not bcl-2 and bcl-X(L) mRNA. These data suggest that aspects of both OPGL's and CSF-1's signaling/survival pathways are required for optimal osteoclast survival. In mice, a single dose of OPG, the OPGL decoy receptor, led to a >90% loss of osteoclasts because of apoptosis within 48 hours of exposure without impacting osteoclast precursor cells. Therefore, OPGL is essential, but not sufficient, for osteoclast survival and endogenous CSF-1 levels are insufficient to maintain osteoclast viability in the absence of OPGL.

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Carrier Proteins / pharmacology*
  • Cell Survival / drug effects*
  • Cells, Cultured
  • Gene Expression Regulation / drug effects
  • Glycoproteins / pharmacology
  • Injections, Subcutaneous
  • Macrophage Colony-Stimulating Factor / pharmacology
  • Male
  • Membrane Glycoproteins / pharmacology*
  • Mice
  • Mice, Inbred C3H
  • NF-kappa B / metabolism
  • Osteoclasts / cytology
  • Osteoclasts / drug effects*
  • Osteoclasts / ultrastructure
  • Osteoprotegerin
  • Proto-Oncogene Proteins c-bcl-2 / genetics
  • RANK Ligand
  • RNA, Messenger / drug effects
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Receptor Activator of Nuclear Factor-kappa B
  • Receptors, Cytoplasmic and Nuclear*
  • Receptors, Tumor Necrosis Factor
  • Time Factors
  • bcl-X Protein

Substances

  • Bcl2l1 protein, mouse
  • Carrier Proteins
  • Glycoproteins
  • Membrane Glycoproteins
  • NF-kappa B
  • Osteoprotegerin
  • Proto-Oncogene Proteins c-bcl-2
  • RANK Ligand
  • RNA, Messenger
  • Receptor Activator of Nuclear Factor-kappa B
  • Receptors, Cytoplasmic and Nuclear
  • Receptors, Tumor Necrosis Factor
  • Tnfrsf11a protein, mouse
  • Tnfrsf11b protein, mouse
  • Tnfsf11 protein, mouse
  • bcl-X Protein
  • Macrophage Colony-Stimulating Factor