Calcium-modulating cyclophilin ligand desensitizes hormone-evoked calcium release

Biochem Biophys Res Commun. 2000 Sep 16;276(1):97-100. doi: 10.1006/bbrc.2000.3442.

Abstract

The Ca(2+)-modulating cyclophilin ligand (CAML) protein causes stimulation of transcription factors via activation of a store-operated Ca(2+) entry pathway. Since CAML is widely expressed in mammalian tissues, it may be an important regulator of Ca(2+) store function. In the present study, we investigated the consequence of CAML overexpression on Ca(2+) signaling using rapid confocal imaging of Fluo3-loaded NIH3T3 fibroblasts. Control and CAML-expressing cells gave concentration-dependent responses to the Ca(2+) mobilizing agonist ATP. CAML expression reduced the sensitivity of the cells so that higher concentrations of ATP were needed to achieve global Ca(2+) waves. The amplitudes of Ca(2+) waves were significantly reduced in CAML expressing cells, consistent with earlier suggestions that CAML causes depletion of internal Ca(2+) stores. With low ATP concentrations, only local Ca(2+) release events were observed. CAML did not affect the characteristics of these local Ca(2+) signals, suggesting that it does not directly affect Ca(2+) release channels.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 3T3 Cells
  • Adaptor Proteins, Signal Transducing*
  • Adenosine Triphosphate / pharmacology*
  • Animals
  • Biological Transport
  • Calcium / physiology*
  • Carrier Proteins / physiology*
  • Dose-Response Relationship, Drug
  • Mice
  • Signal Transduction* / drug effects

Substances

  • Adaptor Proteins, Signal Transducing
  • Caml protein, mouse
  • Carrier Proteins
  • Adenosine Triphosphate
  • Calcium