Potent analgesic effects of GDNF in neuropathic pain states

Science. 2000 Oct 6;290(5489):124-7. doi: 10.1126/science.290.5489.124.

Abstract

Neuropathic pain arises as a debilitating consequence of nerve injury. The etiology of such pain is poorly understood, and existing treatment is largely ineffective. We demonstrate here that glial cell line-derived neurotrophic factor (GDNF) both prevented and reversed sensory abnormalities that developed in neuropathic pain models, without affecting pain-related behavior in normal animals. GDNF reduces ectopic discharges within sensory neurons after nerve injury. This may arise as a consequence of the reversal by GDNF of the injury-induced plasticity of several sodium channel subunits. Together these findings provide a rational basis for the use of GDNF as a therapeutic treatment for neuropathic pain states.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / drug effects
  • Analgesics, Non-Narcotic / pharmacology
  • Analgesics, Non-Narcotic / therapeutic use*
  • Animals
  • Ganglia, Spinal / physiopathology
  • Glial Cell Line-Derived Neurotrophic Factor
  • Hot Temperature
  • Hyperalgesia / drug therapy*
  • Ligation
  • Nerve Fibers / drug effects
  • Nerve Fibers / physiology
  • Nerve Fibers, Myelinated / drug effects
  • Nerve Fibers, Myelinated / physiology
  • Nerve Growth Factors*
  • Nerve Tissue Proteins / pharmacology
  • Nerve Tissue Proteins / therapeutic use*
  • Neural Conduction / drug effects
  • Neurons, Afferent / drug effects
  • Neurons, Afferent / physiology
  • Pain / drug therapy*
  • Pain Threshold / drug effects
  • Peripheral Nervous System Diseases / physiopathology*
  • Rats
  • Reverse Transcriptase Polymerase Chain Reaction
  • Sciatic Nerve
  • Sodium Channels / genetics
  • Sodium Channels / metabolism
  • Spinal Nerves
  • Touch

Substances

  • Analgesics, Non-Narcotic
  • Gdnf protein, rat
  • Glial Cell Line-Derived Neurotrophic Factor
  • Nerve Growth Factors
  • Nerve Tissue Proteins
  • Sodium Channels