ACE-inhibition modulates some endothelial functions in healthy subjects and in normotensive type 1 diabetic patients

Eur J Clin Invest. 2000 Oct;30(10):853-60. doi: 10.1046/j.1365-2362.2000.00721.x.

Abstract

Background: The usefulness of treatment with an angiotensin-converting enzyme-inhibitor (ACE-inhibitor) in normotensive patients with type 1 diabetes is controversial. We investigated whether ACE-inhibition improves endothelial function in such patients and compared the responses to those in healthy subjects.

Design: We studied 23 healthy volunteers (controls, aged 29.8 [SD 7.0] years) and 24 type 1 diabetic patients (aged 28.7 [9. 6] years; HbA1c 8.1 [1.2]%; diabetes duration 13.8 [2-30] years; blood pressure < 140/90 mm Hg; 7 with microalbuminuria) after 5 weeks of ACE-inhibition (quinapril, 10 mg day-1) and placebo in a randomized, double-blind cross-over design. Estimates of endothelial function obtained were by flow-mediated vasodilation and plasma levels of endothelium-derived proteins.

Results: As estimated from the measurements on placebo, type 1 diabetic patients, as compared to the controls, had some impairment of endothelial function: plasma tissue-type plasminogen activator levels were lower (3.5 vs. 5.4 ng mL(-1), P<0.05), but there were no significant differences in brachial artery flow-mediated vasodilation or plasma levels of von Willebrand Factor, endothelin-1, plasminogen activator inhibitor-1, soluble E-selectin or vascular cell adhesion molecule-1. As compared to placebo, ACE-inhibition increased flow-mediated vasodilation in controls (by 3.84% points [95% CI, 0.66 - 7.02], P<0.05), but not in type 1 diabetic patients (0.82% points [95% CI, -2.72 - 4.36], P = 0.64; P = 0.08 vs. controls). On ACE-inhibition soluble E-selectin levels decreased both in controls (from 43.0 to 37.0 ng mL(-1), P<0.01) and in type 1 diabetic patients (from 41.0 to 39.0 ng mL(-1), P = 0.09). Other endothelial markers did not change during ACE-inhibition.

Conclusion: Normotensive type 1 diabetic patients with normoalbuminara or microalbuminuria have mild endothelial dysfunction. Short-term ACE-inhibition improves endothelial function as reflected by a decreased sE-selectin in healthy subjects and in normotensive type 1 diabetic patients. In healthy subjects, ACE-inhibition increases flow-mediated vasodilation. In contrast, in type 1 diabetic patients, ACE-inhibition does not affect flow-mediated vasodilation.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Angiotensin-Converting Enzyme Inhibitors / administration & dosage*
  • Biomarkers
  • Brachial Artery / physiology
  • Cross-Over Studies
  • Diabetes Mellitus, Type 1 / blood
  • Diabetes Mellitus, Type 1 / complications*
  • Diabetic Angiopathies / blood
  • Diabetic Angiopathies / drug therapy*
  • Double-Blind Method
  • E-Selectin / blood
  • Endothelins / blood
  • Endothelium, Vascular / drug effects*
  • Endothelium, Vascular / metabolism
  • Female
  • Humans
  • Isoquinolines / administration & dosage*
  • Male
  • Plasminogen Activator Inhibitor 1 / blood
  • Quinapril
  • Tetrahydroisoquinolines*
  • Tissue Plasminogen Activator / blood
  • Vascular Cell Adhesion Molecule-1 / blood
  • Vasodilation / drug effects
  • von Willebrand Factor / metabolism

Substances

  • Angiotensin-Converting Enzyme Inhibitors
  • Biomarkers
  • E-Selectin
  • Endothelins
  • Isoquinolines
  • Plasminogen Activator Inhibitor 1
  • Tetrahydroisoquinolines
  • Vascular Cell Adhesion Molecule-1
  • von Willebrand Factor
  • Tissue Plasminogen Activator
  • Quinapril