Styrene inhibits monoamine oxidase A, but not monoamine oxidase B in monkey brain mitochondria

Toxicol Lett. 2000 Sep 30;117(1-2):115-9. doi: 10.1016/s0378-4274(00)00241-1.

Abstract

The effects of styrene on mitochondrial monoamine oxidase (MAO) activity in rat and monkey brains were compared in vitro. After preincubation at 25 degrees C for 20 min with 1 mM styrene monomer MAO-A activity in monkey brain was inhibited potently using 5-HT (for MAO-A substrate), but MAO-B activity in monkey brain and platelets were slightly inhibited using beta-PEA (for MAO-B substrate). Styrene monomer also competitively inhibited MAO-A activity in a dose-dependent manner. MAO-A in monkey brain was inhibited by styrene in ascending order of potency: styrene trimer>styrene dimer>styrene monomer. In contrast styrene monomer slightly inhibited both MAO-A and MAO-B activities in rat brain mitochondria. In the present study styrene monomer potently inhibits MAO-A activity, but not MAO-B activity, in monkey brain mitochondria in vitro. These results indicate the inhibiting action of styrene differs depending on animal species and MAO isoforms.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Brain / drug effects*
  • Brain / enzymology
  • Dose-Response Relationship, Drug
  • Kinetics
  • Macaca
  • Male
  • Mitochondria / drug effects*
  • Mitochondria / enzymology
  • Monoamine Oxidase / drug effects*
  • Monoamine Oxidase / metabolism
  • Phenethylamines / metabolism
  • Rats
  • Rats, Wistar
  • Serotonin / metabolism
  • Styrene / pharmacology*
  • Substrate Specificity

Substances

  • Phenethylamines
  • phenethylamine
  • Serotonin
  • Styrene
  • Monoamine Oxidase