Evaluation in the baboon model of (99m)Tc-biguanide as a tracer for renal imaging

Nucl Med Biol. 2000 Aug;27(6):593-7. doi: 10.1016/s0969-8051(00)00128-1.

Abstract

Studies in various animal species have recently shown that (99m)Tc-BIG has practical and dosimetric benefits for renal imaging that could probably make it a good alternative to (99m)Tc-2, 3-dimercaptosuccinic acid ((99m)Tc-DMSA). In this study, using the baboon experimental model, the biodistribution of (99m)Tc-BIG and (99m)Tc-DMSA are compared. It is demonstrated that early good contrast imaging and more favourable dosimetry is possible with (99m)Tc-BIG compared to (99m)Tc-DMSA, confirming the quoted previous findings with small animals. Time-activity curves for kidneys and other organs support these findings, and MIRDOSE software provided the dosimetry.

Publication types

  • Comparative Study
  • Evaluation Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biguanides / pharmacokinetics*
  • Drug Evaluation, Preclinical
  • Heart / diagnostic imaging
  • Kidney / diagnostic imaging*
  • Kidney / metabolism
  • Liver / diagnostic imaging
  • Liver / metabolism
  • Lung / diagnostic imaging
  • Lung / metabolism
  • Male
  • Metabolic Clearance Rate
  • Models, Biological
  • Myocardium / metabolism
  • Papio
  • Radionuclide Imaging
  • Radiopharmaceuticals / pharmacokinetics*
  • Radiotherapy Planning, Computer-Assisted
  • Spleen / diagnostic imaging
  • Spleen / metabolism
  • Technetium Tc 99m Dimercaptosuccinic Acid / pharmacokinetics*
  • Tissue Distribution

Substances

  • Biguanides
  • Radiopharmaceuticals
  • technetium Tc 99m biguanide
  • Technetium Tc 99m Dimercaptosuccinic Acid