Phospholamban decreases the energetic efficiency of the sarcoplasmic reticulum Ca pump

J Biol Chem. 2001 Mar 9;276(10):7195-201. doi: 10.1074/jbc.M007085200. Epub 2000 Nov 21.

Abstract

We tested the hypothesis that increased Sarcoplasmic reticulum (SR) Ca content ([Ca](SRT)) in phospholamban knockout mice (PLB-KO) is because of increased SR Ca pump efficiency defined by the steady-state SR [Ca] gradient. The time course of thapsigargin-sensitive ATP-dependent (45)Ca influx into and efflux out of cardiac SR vesicles from PLB-KO and wild-type (WT) mice was measured at 100 nm free [Ca]. We found that PLB decreased the initial SR Ca uptake rate (0.13 versus 0.31 nmol/mg/s) and decreased steady-state (45)Ca content (0.9 versus 4.1 nmol/mg protein). Furthermore, at similar total SR [Ca], the pump-mediated Ca efflux rate was higher in WT (0.065 versus 0.037 nmol/mg/s). The pump-independent leak rate constant (k(leak)) was also measured at 100 nm free [Ca]. The results indicate that k(leak) was < 1% of pump-mediated backflux and was not different among nonpentameric mutant PLB (PLB-C41F), WT pentameric PLB (same expression level), and PLB-KO. Therefore differences in passive SR Ca leak cannot be the cause of the higher thapsigargin-sensitive Ca efflux from the WT membranes. We conclude that the decreased total SR [Ca] in WT mice is caused by decreased SR Ca influx rate, an increased Ca-pump backflux, and unaltered leak. Based upon both thermodynamic and kinetic analysis, we conclude that PLB decreases the energetic efficiency of the SR Ca pump.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Calcium / pharmacokinetics
  • Calcium-Binding Proteins / metabolism*
  • Calcium-Transporting ATPases / metabolism*
  • Enzyme Inhibitors / metabolism*
  • Kinetics
  • Mice
  • Mice, Knockout
  • Myocardium / cytology*
  • Myocardium / metabolism*
  • Protein Binding
  • Sarcoplasmic Reticulum / metabolism*
  • Thapsigargin / pharmacology
  • Thermodynamics
  • Time Factors

Substances

  • Calcium-Binding Proteins
  • Enzyme Inhibitors
  • phospholamban
  • Thapsigargin
  • Calcium-Transporting ATPases
  • Calcium