The status of voltage-dependent calcium channels in alpha 1E knock-out mice

J Neurosci. 2000 Dec 1;20(23):8566-71. doi: 10.1523/JNEUROSCI.20-23-08566.2000.

Abstract

It has been hypothesized that R-type Ca currents result from the expression of the alpha(1E) gene. To test this hypothesis we examined the properties of voltage-dependent Ca channels in mice in which the alpha(1E) Ca channel subunit had been deleted. Application of omega-conotoxin GVIA, omega-agatoxin IVA, and nimodipine to cultured cerebellar granule neurons from wild-type mice inhibited components of the whole-cell Ba current, leaving a "residual" R current with an amplitude of approximately 30% of the total Ba current. A minor portion of this R current was inhibited by the alpha(1E)-selective toxin SNX-482, indicating that it resulted from the expression of alpha(1E). However, the majority of the R current was not inhibited by SNX-482. The SNX-482-sensitive portion of the granule cell R current was absent from alpha(1E) knock-out mice. We also identified a subpopulation of dorsal root ganglion (DRG) neurons from wild-type mice that expressed an SNX-482-sensitive component of the R current. However as with granule cells, most of the DRG R current was not blocked by SNX-482. We conclude that there exists a component of the R current that results from the expression of the alpha(1E) Ca channel subunit but that the majority of R currents must result from the expression of other Ca channel alpha subunits.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Barium / pharmacology
  • Blotting, Western
  • Calcium / metabolism
  • Calcium Channel Blockers / pharmacology
  • Calcium Channels, R-Type / drug effects
  • Calcium Channels, R-Type / genetics*
  • Calcium Channels, R-Type / metabolism*
  • Cell Survival / genetics
  • Cells, Cultured
  • Cerebellum / cytology
  • Cerebellum / drug effects
  • Cerebellum / metabolism
  • Electrophysiology
  • Ganglia, Spinal / cytology
  • Ganglia, Spinal / drug effects
  • Ganglia, Spinal / metabolism
  • Ion Transport / drug effects
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Neurons / cytology
  • Neurons / drug effects
  • Neurons / metabolism
  • Nimodipine / pharmacology
  • Patch-Clamp Techniques
  • Protein Subunits
  • Spider Venoms / pharmacology
  • Synaptic Transmission / drug effects
  • omega-Agatoxin IVA / pharmacology
  • omega-Conotoxin GVIA / pharmacology

Substances

  • Calcium Channel Blockers
  • Calcium Channels, R-Type
  • Protein Subunits
  • SNX 482
  • Spider Venoms
  • omega-Agatoxin IVA
  • Barium
  • Nimodipine
  • omega-Conotoxin GVIA
  • Calcium