Inhibition of tumor growth in a human neuroblastoma xenograft model with TNP-470

Med Pediatr Oncol. 2000 Dec;35(6):673-6. doi: 10.1002/1096-911x(20001201)35:6<673::aid-mpo41>3.0.co;2-o.

Abstract

Background and Procedure High-risk neuroblastoma disease features are correlated with tumor vascularity, suggesting that angiogenesis inhibitors may be a useful addition to current therapeutic strategies. We therefore examined the efficacy of TNP-470 (TAP Pharmaceuticals, Deerfield, IL) in human neuroblastoma xenograft models.

Results: Tumor growth rate was markedly inhibited in mice receiving TNP-470 administered alone with a treatment to control ratio (T/C) at day 21 = 0.4 (P <.001). TNP-470 also significantly inhibited tumorigenicity when administered shortly after xenograft inoculation (T/C at day 30 = 0.1, P <.001) and when administered following cyclophosphamide (T/C at day 35 = 0.1, P <.001).

Conclusions: These data show that TNP-470 is a potent inhibitor of human neuroblastoma growth both alone and when given with conventional chemotherapy, suggesting that it may be a useful adjunctive therapy for high-risk neuroblastoma patients.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiogenesis Inhibitors / therapeutic use*
  • Animals
  • Child
  • Cyclohexanes
  • Humans
  • Mice
  • Mice, Nude
  • Neoplasm, Residual
  • Neuroblastoma / drug therapy*
  • O-(Chloroacetylcarbamoyl)fumagillol
  • Sesquiterpenes / therapeutic use*
  • Tumor Cells, Cultured
  • Xenograft Model Antitumor Assays

Substances

  • Angiogenesis Inhibitors
  • Cyclohexanes
  • Sesquiterpenes
  • O-(Chloroacetylcarbamoyl)fumagillol