Intramuscular administration of estrogen may promote angiogenesis and perfusion in a rabbit model of chronic limb ischemia

Cardiovasc Res. 2001 Feb 16;49(3):626-33. doi: 10.1016/s0008-6363(00)00199-1.

Abstract

Objective: Promoting angiogenesis may be an effective treatment for patients with diffuse peripheral vascular disease. This study investigated whether estrogen can promote angiogenesis and perfusion in a rabbit model of chronic limb ischemia.

Methods and results: Ischemia was induced in one hindlimb of 24 oophorectomized New Zealand White rabbits. Ten days later (day 0), they were randomized into 4 groups for intramuscular treatment in the ischemic limb: controls receiving saline at day 0; Estrogen-1 group receiving estradiol valerate, modified release (EVMR), 1 mg/kg at day 0; Estrogen-2 group receiving EVMR 1 mg/kg at days 0 and 15; and Estrogen-3 group receiving EVMR 2 mg/kg at day 0. Revascularization was evaluated by clinical indexes, such as ischemic/normal limb systolic blood pressure (BPR), and capillary density/muscle fiber in the abductor muscle of the ischemic limb at the time of death (day 30). At day 30 the BPR was increased in all groups (0.39+/-0.08 in the controls, 0.52+/-0.11 in the Estrogen-1 group, 0.65+/-0.13 in the Estrogen-2 group and 0.61+/-0.16 in the Estrogen-3 group, F=2.39, P=0.04). The capillary/muscle fiber at day 30 was 0.87+/-0.09, 1.08+/-0.15, 1.01+/-0.14 and 1.10+/-0.9 (F=5.01, P=0.01), respectively, in the 4 groups. The capillary/muscle fiber was related to BPR (r=0.48, P<0.02) and to 17-beta estradiol plasma levels of day 15 (r=0.58, P=0.003) and of day 30 (r=0.46, P<0.02).

Conclusion: Administration of estrogen promotes angiogenesis and perfusion in ischemic rabbit hindlimbs. Thus, estrogen may represent a new therapeutic modality in the management of arterial insufficiency.

MeSH terms

  • Animals
  • Blood Pressure / drug effects
  • Capillaries
  • Collateral Circulation*
  • Delayed-Action Preparations
  • Drug Administration Schedule
  • Estradiol / administration & dosage*
  • Estradiol / blood
  • Female
  • Hindlimb / blood supply*
  • Injections, Intramuscular
  • Ischemia / physiopathology
  • Ischemia / therapy*
  • Laser-Doppler Flowmetry
  • Muscle Fibers, Skeletal / drug effects
  • Neovascularization, Physiologic*
  • Ovariectomy
  • Perfusion
  • Rabbits
  • Random Allocation
  • Regression Analysis

Substances

  • Delayed-Action Preparations
  • Estradiol