Coenzyme Q protects cells against serum withdrawal-induced apoptosis by inhibition of ceramide release and caspase-3 activation

Antioxid Redox Signal. 2000 Summer;2(2):263-75. doi: 10.1089/ars.2000.2.2-263.

Abstract

Coenzyme Q10 (CoQ10) is a component of the antioxidant machinery that protects cell membranes from oxidative damage and decreases apoptosis in leukemic cells cultured in serum-depleted media. Serum deprivation induced apoptosis in CEM-C7H2 (CEM) and to a lesser extent in CEM-9F3, a subline overexpressing Bcl-2. Addition of CoQ10 to serum-free media decreased apoptosis in both cell lines. Serum withdrawal induced an early increase of neutral-sphingomyelinase activity, release of ceramide, and activation of caspase-3 in both cell lines, but this effect was more pronounced in CEM cells. CoQ10 prevented activation of this cascade of events. Lipids extracted from serum-depleted cultures activated caspase-3 independently of the presence of mitochondria in cell-free in vitro assays. Activation of caspase-3 by lipid extracts or ceramide was prevented by okadaic acid, indicating the implication of a phosphatase in this process. Our results support the hypothesis that plasma membrane CoQ10 regulate the initiation phase of serum withdrawal-induced apoptosis by preventing oxidative damage and thus avoiding activation of downstream effectors as neutral-sphingomyelinase and subsequent ceramide release and caspase activation pathways.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis*
  • Caspase 3
  • Caspase Inhibitors*
  • Cell Membrane / metabolism
  • Cell-Free System
  • Ceramides / antagonists & inhibitors*
  • Coenzymes
  • Culture Media, Serum-Free
  • Electron Transport Complex IV / metabolism
  • Enzyme Activation / drug effects
  • Humans
  • Leukemia / metabolism
  • Lipid Metabolism
  • Mitochondria / metabolism
  • Okadaic Acid / metabolism
  • Oxidative Stress
  • Sphingomyelin Phosphodiesterase / metabolism
  • Time Factors
  • Tumor Cells, Cultured
  • Ubiquinone / analogs & derivatives
  • Ubiquinone / metabolism*

Substances

  • Caspase Inhibitors
  • Ceramides
  • Coenzymes
  • Culture Media, Serum-Free
  • Ubiquinone
  • Okadaic Acid
  • Electron Transport Complex IV
  • Sphingomyelin Phosphodiesterase
  • CASP3 protein, human
  • Caspase 3
  • coenzyme Q10