Effect of FR167653 on pancreatic ischemia-reperfusion injury in dogs

Surgery. 2001 Mar;129(3):309-17. doi: 10.1067/msy.2001.111193.

Abstract

Background: The role of inflammatory cytokines is still unclear in ischemia-reperfusion injury of the pancreas. We investigated the effect of FR167653 (FR), a newly developed compound that is a potent suppressor of interleukin (IL)-1beta and tumor necrosis factor (TNF)-alpha on ischemia-reperfusion injury of the isolated pancreatic tail in dogs.

Methods: The tail of the pancreas was subjected to ischemia for 90 minutes. During occlusion of the vascular inflow, the head of the pancreas was removed. A control group (n = 14) and an FR treatment group (n = 11) were evaluated for survival rate, tissue blood flow, arterial oxygen pressure (Pao(2)), serum amylase and lipase levels, glucose and insulin, liver enzymes, creatinine, IL-1beta mRNA in the peripheral blood, and histopathology.

Results: Six of the 14 control animals and 2 of the 11 FR-treated animals died. The FR treatment group showed lower amylase (P=.037) and lipase (P =.030) levels, lower IL-1beta mRNA expression (P =.033), and less pancreatic tissue damage (P =.041) than did the control group, but there was no remarkable change in endocrine function (P =.422). Pao(2) during the acute phase in the FR treatment group was maintained (P=.009), but pulmonary tissue was damaged. Results of biochemical and histologic examinations of the liver and kidneys were unremarkable.

Conclusions: FR ameliorates ischemia-reperfusion injury of the pancreas and reduces the production of inflammatory cytokines that may contribute to secondary damage to distant organs.

MeSH terms

  • Animals
  • Dogs
  • Female
  • Interleukin-1 / blood
  • Ischemia / pathology*
  • Ischemia / physiopathology*
  • Islets of Langerhans / physiopathology
  • Male
  • Pancreas / blood supply*
  • Pancreas / physiopathology
  • Pyrazoles / pharmacology*
  • Pyridines / pharmacology*
  • Reperfusion Injury / pathology*
  • Reperfusion Injury / physiopathology*

Substances

  • FR 167653
  • Interleukin-1
  • Pyrazoles
  • Pyridines