Structure of an extracellular gp130 cytokine receptor signaling complex

Science. 2001 Mar 16;291(5511):2150-5. doi: 10.1126/science.1058308.

Abstract

The activation of gp130, a shared signal-transducing receptor for a family of cytokines, is initiated by recognition of ligand followed by oligomerization into a higher order signaling complex. Kaposi's sarcoma-associated herpesvirus encodes a functional homolog of human interleukin-6 (IL-6) that activates human gp130. In the 2.4 angstrom crystal structure of the extracellular signaling assembly between viral IL-6 and human gp130, two complexes are cross-linked into a tetramer through direct interactions between the immunoglobulin domain of gp130 and site III of viral IL-6, which is necessary for receptor activation. Unlike human IL-6 (which uses many hydrophilic residues), the viral cytokine largely uses hydrophobic amino acids to contact gp130, which enhances the complementarity of the viral IL-6-gp130 binding interfaces. The cross-reactivity of gp130 is apparently due to a chemical plasticity evident in the amphipathic gp130 cytokine-binding sites.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Antigens, CD / chemistry*
  • Antigens, CD / metabolism*
  • Binding Sites
  • Crystallization
  • Crystallography, X-Ray
  • Cytokine Receptor gp130
  • Epitopes
  • Humans
  • Hydrogen Bonding
  • Interleukin-6 / chemistry*
  • Interleukin-6 / immunology
  • Interleukin-6 / metabolism*
  • Membrane Glycoproteins / chemistry*
  • Membrane Glycoproteins / metabolism*
  • Models, Molecular
  • Molecular Mimicry
  • Protein Conformation
  • Protein Structure, Quaternary
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Signal Transduction
  • Viral Proteins / chemistry*
  • Viral Proteins / immunology
  • Viral Proteins / metabolism*

Substances

  • Antigens, CD
  • Epitopes
  • IL6ST protein, human
  • Interleukin-6
  • Membrane Glycoproteins
  • Viral Proteins
  • Cytokine Receptor gp130

Associated data

  • PDB/1I1R