Effects of epidermal growth factor on CYP inducibility by xenobiotics, DNA replication, and caspase activations in collagen I gel sandwich cultures of rat hepatocytes

Biochem Pharmacol. 2001 May 15;61(10):1293-303. doi: 10.1016/s0006-2952(01)00612-8.

Abstract

In this study, we investigated the combined effects of EGF and collagen I gel on the phenotype of cultured rat hepatocytes and we focussed our investigations on the regulation of xenobiotic-mediated induction of CYP, cell cycle progression and activation of capases 8 and 3. We found that EGF, added to basal culture medium or phenobarbital (3.2 mM) containing medium, provoked a moderate decrease of CYP1A1 and CYP2B1/2 activities. However, EGF did not exert any inhibitory effect on 3-methylcholantrene (5 microM) and beta-naphtoflavone (25 microM) induction of CYP1A1 activities. In collagen gel sandwich cultures, hepatocytes remained arrested in mid-G1 phase of the cell cycle, even in the presence of EGF. In conventional primary cultures, caspases 8 and 3 were activated at 3 and 5 days after plating respectively. In collagen gel sandwich cultures, we found that neither collagen I nor EGF prevented activation of caspase 8 while collagen I gel inhibited activation of caspase 3, preventing spontaneous apoptosis of cultured rat hepatocytes. In contrast, EGF transiently increased caspase 3 activity at day 1 after plating. Altogether, our data demonstrate that collagen I gel triggers intracellular signals which strongly affect cultured hepatocyte phenotype, leading to a cell cycle arrest in G1 phase and long-term survival through the inhibition of caspase 3 activation and that EGF-free medium improves survival and liver-specific gene expression in hepatocytes maintained in collagen I gel sandwich cultures.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Caspase 3
  • Caspases / metabolism*
  • Cell Cycle / drug effects
  • Cell Survival / drug effects
  • Collagen / pharmacology
  • Cytochrome P-450 CYP1A1 / drug effects
  • Cytochrome P-450 CYP1A1 / metabolism*
  • Cytochrome P-450 CYP2B1 / drug effects
  • Cytochrome P-450 CYP2B1 / metabolism*
  • DNA Replication / drug effects
  • Drug Interactions
  • Enzyme Activation
  • Enzyme Induction / drug effects
  • Epidermal Growth Factor / pharmacology*
  • Hepatocytes / drug effects*
  • Hepatocytes / enzymology
  • In Vitro Techniques
  • Male
  • Rats
  • Rats, Sprague-Dawley
  • Serum Albumin / metabolism
  • Xenobiotics / pharmacology*

Substances

  • Serum Albumin
  • Xenobiotics
  • Epidermal Growth Factor
  • Collagen
  • Cytochrome P-450 CYP1A1
  • Cytochrome P-450 CYP2B1
  • Casp3 protein, rat
  • Caspase 3
  • Caspases