[Effects of 17 beta-estradiol on delayed rectifier potassium channels in hippocampal pyramidal neurons of the rat]

Sheng Li Xue Bao. 1998 Oct;50(5):581-6.
[Article in Chinese]

Abstract

In the present study, both cell-attached and inside-out patch-clamp techniques were used to detect the effects of 17 beta-estradiol (E2) on 42 pS delayed rectifier potassium channels in acutely dissociated hippocampal neurons of new-born SD rats. The results indicated that after application of 1.0 and 10.0 nmol/L E2, the open probabilities of K+ channels were decreased from (67.4 +/- 18.2)% to (41.2 +/- 12.5)% and from (56.3 +/- 15.8)% to (13.2 +/- 12.6)% respectively, the open frequencies were reduced from (43.40 +/- 6.7) Hz to (27.68 +/- 9.1) Hz and from (38.19 +/- 10.1) Hz to (15.79 +/- 3.5) Hz respectively. Meanwhile, there was a shortening of the mean open time and a lenghtening of the mean close time of the channels. The above results suggest that E2 has suppressive effects on the activities of the channels, which might be exerted through a direct action on the cellular membrane.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biological Transport, Active
  • Delayed Rectifier Potassium Channels
  • Electrophysiology
  • Estradiol / pharmacology*
  • Female
  • Hippocampus / physiology*
  • In Vitro Techniques
  • Male
  • Neurons / physiology
  • Patch-Clamp Techniques
  • Potassium / metabolism*
  • Potassium Channels / drug effects*
  • Potassium Channels, Voltage-Gated*
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Delayed Rectifier Potassium Channels
  • Potassium Channels
  • Potassium Channels, Voltage-Gated
  • Estradiol
  • Potassium