The snake venom toxin alboaggregin-A activates glycoprotein VI

Blood. 2001 Jun 15;97(12):3989-91. doi: 10.1182/blood.v97.12.3989.

Abstract

The glycoprotein (GP)-Ib-IX-V receptor complex has recently been reported to signal through a pathway similar to that used by the collagen receptor GPVI, with a critical role described for the Fc receptor gamma-chain. The evidence for this was based in part on studies with the GPIbalpha-selective snake venom toxin, alboaggregin-A. In the present study, it is reported that alboaggregin-A has activity at the collagen receptor GPVI in addition to GPIbalpha, and evidence is provided that this contributes to protein tyrosine phosphorylation, shape change, and GPIIb-IIIa-dependent aggregation. This may explain why responses to alboaggregin-A are distinct from those to von Willebrand factor-ristocetin. (Blood. 2001;97:3989-3991)

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blood Platelets / cytology
  • Blood Platelets / drug effects
  • Crotalid Venoms / metabolism
  • Crotalid Venoms / pharmacology*
  • Humans
  • Phosphorylation / drug effects
  • Platelet Aggregation / drug effects
  • Platelet Glycoprotein GPIIb-IIIa Complex / pharmacology
  • Platelet Membrane Glycoproteins / drug effects*
  • Platelet Membrane Glycoproteins / metabolism
  • Platelet Membrane Glycoproteins / physiology
  • Signal Transduction / drug effects
  • Tyrosine / metabolism

Substances

  • Crotalid Venoms
  • Platelet Glycoprotein GPIIb-IIIa Complex
  • Platelet Membrane Glycoproteins
  • alboaggregin A
  • platelet membrane glycoprotein VI
  • Tyrosine