Controlling tumor-derived and vascular endothelial cell growth: role of the 4Ff2 cell surface antigen

Am J Pathol. 2001 Jul;159(1):165-78. doi: 10.1016/s0002-9440(10)61683-5.

Abstract

We have isolated a monoclonal antibody, clone betaE11, which recognizes an antigen that is highly abundant on the surface of mitotic vascular endothelial cells and tumor cells. By sodium dodecyl sulfate-polyacrylamide gel electrophoresis and Western blotting, expression of this 190-kd antigen is approximately threefold higher in mitotic versus interphase endothelial cells. Treatment of tumor cells with an antibody to the betaE11 antigen inhibits their growth in a dose-dependent manner in vitro with maximal inhibition at an antibody concentration of 1 microg/ml. Different tumor cell lines demonstrate varying sensitivities to anti-betaE11 with the following order of growth inhibition: colon > prostate = glioma > melanoma = fibroblast > breast > liver. Furthermore, the betaE11 antigen localizes to regions of prostatic intraductal neoplasia in paraffin-embedded sections. Mass spectrometry of the cell-derived betaE11 protein and V8-protease fingerprint analysis indicate that the betaE11 antigen is nearly identical to the 4F2 heavy chain antigen, a cell surface protein that has been implicated in cell activation and proliferation. Expression of the betaE11 antigen during mitosis functionally links it to a fundamental aspect of cell proliferation, and its spatial localization on the surface of both proliferating endothelium and tumor cells demonstrates its potential for tumor immunotherapy.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies / pharmacology
  • Antigens, CD / chemistry
  • Antigens, CD / physiology*
  • Antigens, Surface / chemistry
  • Antigens, Surface / immunology
  • Antigens, Surface / metabolism
  • Blotting, Western
  • Carrier Proteins / chemistry
  • Carrier Proteins / physiology*
  • Cattle
  • Cell Division / drug effects
  • Cell Division / physiology
  • Cells, Cultured
  • Endothelium, Vascular / cytology*
  • Endothelium, Vascular / metabolism
  • Fusion Regulatory Protein-1
  • Glycosylation
  • Mitosis / physiology
  • Neoplasms / metabolism
  • Neoplasms / pathology*
  • Protein Processing, Post-Translational
  • Tissue Distribution

Substances

  • Antibodies
  • Antigens, CD
  • Antigens, Surface
  • Carrier Proteins
  • Fusion Regulatory Protein-1
  • betaE11 antigen, bovine