Inhibition of ERalpha-mediated trans-activation of human coagulation factor XII gene by heteromeric transcription factor NF-Y

Endocrinology. 2001 Aug;142(8):3380-8. doi: 10.1210/endo.142.8.8345.

Abstract

Human coagulation factor XII promoter contains an estrogen response element that mediates ligand-activated ERalpha induction of coagulation factor XII gene expression. The 3'-half of coagulation factor XII-estrogen response element overlaps a putative CCAAT box, the widespread regulatory element specifically recognized by the heteromeric transcription factor NF-Y. Transient cotransfection of NF-Y and ERalpha results in strong inhibition of estrogen stimulation of coagulation factor XII promoter activity. NF-Y antagonism is primarily exerted by the NF-YA subunit and does not require binding to the CCAAT element, as NF-YA mutants with impaired DNA binding capacity retain the ability to inhibit ERalpha trans-activation. EMSAs with increasing concentrations of recombinant NF-Y do not detect the formation of NF-Y-DNA complexes or show impairment of ERalpha binding to estrogen response element. Immunoprecipitation of whole cell extracts with anti-ERalpha antibody reveals an in vivo association between the two transcription factors, which is abolished by deletion of the NF-YA carboxyl-terminus. In functional experiments with sequential NF-YA deletion mutants the HAP2-homology region appears essential in eliciting NF-YA antagonistic activity. In conclusion, our results demonstrate that heteromeric transcription factor NF-Y inhibits estrogen induction of coagulation factor XII promoter in a DNA binding-independent fashion and suggest a novel role for NF-Y as a partner for the ERalpha transcription complex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3 Cells
  • Animals
  • Base Sequence / genetics
  • CCAAT-Binding Factor / genetics
  • CCAAT-Binding Factor / pharmacology
  • CCAAT-Binding Factor / physiology*
  • DNA / metabolism
  • Estradiol / pharmacology
  • Estrogen Receptor alpha
  • Factor XII / genetics*
  • Gene Expression Regulation / drug effects
  • Humans
  • Mice
  • Molecular Sequence Data
  • Promoter Regions, Genetic / drug effects
  • Protein Isoforms / genetics
  • Protein Isoforms / pharmacology
  • Protein Structure, Tertiary / genetics
  • Receptors, Estrogen / physiology*
  • Transcription, Genetic / drug effects
  • Transcriptional Activation / physiology*
  • Tumor Cells, Cultured

Substances

  • CCAAT-Binding Factor
  • Estrogen Receptor alpha
  • Protein Isoforms
  • Receptors, Estrogen
  • Estradiol
  • Factor XII
  • DNA