Radiation-induced glomerular thrombus formation and nephropathy are not prevented by the ADP receptor antagonist clopidogrel

Int J Radiat Oncol Biol Phys. 2001 Aug 1;50(5):1332-8. doi: 10.1016/s0360-3016(01)01617-0.

Abstract

Purpose: To assess the effects of kidney irradiation on glomerular adenosine diphosphatase (ADPase) activity and intraglomerular microthrombus formation, and their correlation to the development of renal functional impairment.

Methods and materials: C3H/HenAf-nu(+) mice were given single-dose or fractionated kidney irradiations. Glomerular ADPase activity was measured using a cerium-based histochemical method. Microthrombus formation within the glomeruli was assessed by a semiquantitative immunohistochemical analysis of fibrinogen/fibrin deposits. Renal function was assessed by the [(51)Cr]EDTA retention assay.

Results: The ADPase activity was significantly reduced, to approximately 50% of pretreatment value, 4--40 weeks after 10--16 Gy single-dose irradiation and at 44 weeks after 20 x 2 Gy. No dose--effect relationship was found. An approximately fourfold increase in glomerular fibrinogen/fibrin staining was observed at 1 year after irradiation. This increase was not influenced by treating the mice with daily, oral clopidogrel, a platelet ADP receptor antagonist, which reduced platelet aggregation by more than 75%. Radiation-induced impairment of glomerular filtration was also not affected by the clopidogrel treatment.

Conclusion: These data indicate that irradiation significantly reduced glomerular ADPase activity, which correlated with an increased glomerular fibrinogen/fibrin deposition. We were not able to reduce these prothrombotic changes, nor to protect against radiation nephropathy, by pharmacological intervention with an ADP-receptor antagonist.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apyrase / antagonists & inhibitors*
  • Clopidogrel
  • Dose Fractionation, Radiation
  • Dose-Response Relationship, Radiation
  • Drug Evaluation, Preclinical
  • Edetic Acid / pharmacokinetics
  • Female
  • Fibrin Fibrinogen Degradation Products / analysis
  • Fibrinolytic Agents / therapeutic use*
  • Glomerular Filtration Rate / radiation effects
  • Image Processing, Computer-Assisted
  • Kidney Function Tests
  • Kidney Glomerulus / radiation effects*
  • Mice
  • Mice, Inbred C3H
  • Mice, Nude
  • Purinergic P2 Receptor Antagonists*
  • Radiation Injuries, Experimental / drug therapy
  • Radiation Injuries, Experimental / prevention & control*
  • Radiation Tolerance
  • Thrombosis / drug therapy
  • Thrombosis / etiology
  • Thrombosis / prevention & control*
  • Ticlopidine / analogs & derivatives
  • Ticlopidine / therapeutic use*

Substances

  • Fibrin Fibrinogen Degradation Products
  • Fibrinolytic Agents
  • Purinergic P2 Receptor Antagonists
  • Edetic Acid
  • Clopidogrel
  • Apyrase
  • Ticlopidine