Preparation and properties of an alpha-1-protease inhibitor concentrate with high specific activity

Vox Sang. 2001 Jul;81(1):29-36. doi: 10.1046/j.1423-0410.2001.00049.x.

Abstract

Background and objectives: Because the current demand for alpha-1-protease inhibitor (A1PI) exceeds the available supply, we aimed to develop a process for purification of A1PI from plasma which would achieve the highest possible degree of purity, specific activity and yield.

Materials and methods: A1PI was purified from Cohn fraction IV-1,4 using ethanol precipitation and Q-Sepharose chromatography. Ceramic hydroxyapatite chromatography was used as a final purification step. Two independent virus-inactivation procedures (chemical and vapour heating) were applied.

Results: The resulting A1PI had an unprecedented high specific activity. In addition, the process led to the discovery of a new isoform of A1PI in isoelectric focusing gels.

Conclusion: The high specific activity of the A1PI preparation achieved with this process should allow a reduction of the A1PI total protein load necessary to achieve clinically relevant effects.

Publication types

  • Comparative Study

MeSH terms

  • Blood Proteins / chemistry
  • Chemical Precipitation
  • Chromatography, Agarose
  • Humans
  • Isoelectric Focusing
  • Pancreatic Elastase / antagonists & inhibitors
  • Protein Isoforms
  • Serine Proteinase Inhibitors / isolation & purification
  • Serine Proteinase Inhibitors / pharmacology
  • Serine Proteinase Inhibitors / standards
  • Sterilization
  • Therapeutic Equivalency
  • Trypsin Inhibitors / isolation & purification
  • Trypsin Inhibitors / pharmacology
  • Trypsin Inhibitors / standards
  • alpha 1-Antitrypsin / isolation & purification*
  • alpha 1-Antitrypsin / pharmacology
  • alpha 1-Antitrypsin / standards*

Substances

  • Blood Proteins
  • Cohn fraction IV
  • Protein Isoforms
  • Serine Proteinase Inhibitors
  • Trypsin Inhibitors
  • alpha 1-Antitrypsin
  • Pancreatic Elastase