Presynaptic modulation by group III metabotropic glutamate receptors (mGluRs) of the excitatory postsynaptic potential mediated by mGluR1 in rat cerebellar Purkinje cells

Neurosci Lett. 2001 Sep 7;310(1):61-5. doi: 10.1016/s0304-3940(01)02082-1.

Abstract

Purkinje neurons were recorded from rat cerebellar slices. Parallel fibres stimulation elicited a fast excitatory postsynaptic potential (EPSP) mediated by ionotropic glutamate (iGluR) -amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors followed by the inhibitory gamma-aminobutyric acidA (GABAA)-dependent postsynaptic potential. In the presence of antagonists for iGluRs and for GABAA receptors, brief tetanic activation evoked a slow metabotropic glutamate receptor (mGluR)-dependent EPSP (mGluR-EPSP). This mGluR-EPSP was blocked by the selective mGluR1 antagonists LY367385 and CPCCOEt, but not by the mGluR5 antagonist MPEP. Group II agonists affected neither iGluR-EPSP nor mGluR-EPSP. Conversely, L-AP4 and L-SOP, group III mGluR agonists, inhibited both iGluR- and mGluR-EPSPs. The depolarisations evoked by both AMPA and group I agonists were unaffected, indicating a presynaptic action of group III mGluRs. These data suggest that glutamate released by parallel fibres activates group III mGluR autoreceptors, depressing both iGluR- and mGluR1-mediated EPSPs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzoates*
  • Bicuculline / pharmacology
  • Cerebellum / physiology*
  • Electric Stimulation
  • Excitatory Amino Acid Antagonists / pharmacology
  • Excitatory Postsynaptic Potentials / physiology*
  • GABA Antagonists / pharmacology
  • Glycine / analogs & derivatives
  • Glycine / pharmacology
  • Male
  • Purkinje Cells / metabolism*
  • Quinoxalines / pharmacology
  • Rats
  • Rats, Wistar
  • Receptors, Metabotropic Glutamate / physiology*
  • Receptors, Presynaptic / physiology*

Substances

  • Benzoates
  • Excitatory Amino Acid Antagonists
  • GABA Antagonists
  • Quinoxalines
  • Receptors, Metabotropic Glutamate
  • Receptors, Presynaptic
  • metabotropic glutamate receptor type 1
  • 2,3-dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline
  • alpha-methyl-4-carboxyphenylglycine
  • Glycine
  • Bicuculline