Effect of ethanol on tracheal potassium channels reconstituted into bilayer lipid membranes

Physiol Res. 2001;50(5):507-11.

Abstract

We examined the effect of ethanol on single potassium channels derived from plasma membranes of bovine tracheal smooth muscles. The observed potassium channels had a conductance of 296 +/- 31 pS (mean +/- S.D.) in symmetrical 250 mmol/l KCl solutions, and exhibited a voltage- and Ca2+-dependence similar to BKCa channels. Ethanol at 50, 100 and 200 mM concentrations increased the probability of open potassium channels to 112 +/- 5, 127 +/- 7 and 121 +/- 13% (mean +/- S.E.M.), respectively. It is suggested that increased activity of the BKCa channels by ethanol hyperpolarizes the plasma membrane and thus may contribute to relaxation of tracheal smooth muscle.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium / pharmacology
  • Cattle
  • Cell Membrane / chemistry
  • Cell Membrane / physiology
  • Electric Conductivity
  • Ethanol / pharmacology*
  • Ion Channel Gating / drug effects
  • Lipid Bilayers / metabolism*
  • Potassium Channels / drug effects*
  • Potassium Channels / physiology*
  • Potassium Chloride / pharmacology
  • Trachea / chemistry*
  • Trachea / physiology

Substances

  • Lipid Bilayers
  • Potassium Channels
  • Ethanol
  • Potassium Chloride
  • Calcium