Induction of the IL-13 receptor alpha2-chain by IL-4 and IL-13 in human keratinocytes: involvement of STAT6, ERK and p38 MAPK pathways

Oncogene. 2001 Oct 11;20(46):6660-8. doi: 10.1038/sj.onc.1204629.

Abstract

IL-4 and IL-13 are related cytokines which induce both pro- and anti-inflammatory effects depending on the cell type they act upon and the nature of the receptors expressed. The type I receptor complex is composed of the IL-4Ralpha and gammac and only binds IL-4, whereas, in the type II receptor, IL-4Ralpha dimerizes with IL-13Ralpha1 upon either IL-4 or IL-13 binding. Another ligand binding chain potentially implicated in the IL-4/IL-13 receptor has been described, the IL-13Ralpha2, but the regulation of its expression and its role in IL-4/IL-13 transduction is poorly understood. In this study we report that IL-4 and IL-13 upregulate IL-13Ralpha2 at both the mRNA and protein levels in the keratinocyte cell line HaCaT. In these cells, IL-4 or IL-13 were shown to activate the Janus Kinases JAK1 and JAK2, the transcription factor STAT6, and the ERK and p38 mitogen-activated protein kinases. We show that IL-4 or IL-13-induced IL-13Ralpha2 mRNA expression was inhibited by the ERK inhibitor U0126, the JAK inhibitor AG490 and, to a lesser extent, the p38 MAPK inhibitor SB203580. Moreover, expression of a constitutive active mutant of STAT6 alone did not modify IL-13Ralpha2 mRNA expression, but potentiated the effects of IL-4 or IL-13 on IL-13Ralpha2 expression. The constitutive active mutants of MEK1 or MKK6 increased the level of expression of IL-13Ralpha2 mRNA even in absence of stimulation. Our findings demonstrate, for the first time, that IL-4 and IL-13 can induce IL-13Ralpha2 expression in keratinocytes, and that the ERK and p38 MAPK together with JAK2 and STAT6 play a critical role in this process.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / pharmacology
  • Blotting, Western
  • Butadienes / pharmacology
  • Cross-Linking Reagents / pharmacology
  • Enzyme Inhibitors / pharmacology
  • Gene Expression Regulation, Neoplastic*
  • Imidazoles / pharmacology
  • Interleukin-13 / metabolism*
  • Interleukin-13 Receptor alpha1 Subunit
  • Interleukin-4 / metabolism*
  • Keratinocytes / metabolism*
  • Kinetics
  • Ligands
  • Mitogen-Activated Protein Kinases / metabolism*
  • Nitriles / pharmacology
  • Plasmids / metabolism
  • Precipitin Tests
  • Protein Binding
  • Pyridines / pharmacology
  • RNA, Messenger / metabolism
  • Receptors, Interleukin / genetics*
  • Receptors, Interleukin / metabolism*
  • Receptors, Interleukin-13
  • Reverse Transcriptase Polymerase Chain Reaction
  • STAT6 Transcription Factor
  • Signal Transduction
  • Time Factors
  • Trans-Activators / metabolism*
  • Transcription, Genetic
  • Tumor Cells, Cultured
  • Tyrphostins / pharmacology
  • p38 Mitogen-Activated Protein Kinases

Substances

  • Antineoplastic Agents
  • Butadienes
  • Cross-Linking Reagents
  • Enzyme Inhibitors
  • IL13RA1 protein, human
  • Imidazoles
  • Interleukin-13
  • Interleukin-13 Receptor alpha1 Subunit
  • Ligands
  • Nitriles
  • Pyridines
  • RNA, Messenger
  • Receptors, Interleukin
  • Receptors, Interleukin-13
  • STAT6 Transcription Factor
  • Trans-Activators
  • Tyrphostins
  • U 0126
  • alpha-cyano-(3,4-dihydroxy)-N-benzylcinnamide
  • Interleukin-4
  • Mitogen-Activated Protein Kinases
  • p38 Mitogen-Activated Protein Kinases
  • SB 203580