The transcriptional factor Tcf-4 contains different binding sites for beta-catenin and plakoglobin

J Biol Chem. 2002 Jan 18;277(3):1884-91. doi: 10.1074/jbc.M110248200. Epub 2001 Nov 15.

Abstract

beta-Catenin and plakoglobin are two related armadillo proteins necessary for the establishment of adhesion junctions and desmosomes. Moreover, beta-catenin can also act as a transcriptional co-activator through its interaction with the members of Tcf/LEF-1 transcriptional factor family. We show here that Tcf-4 can be phosphorylated in vitro by protein kinase CK2 stoichiometrically in amino acids Ser-58-Ser-59-Ser-60. Phosphorylation of these residues does not modify the interaction of Tcf-4 with beta-catenin but reduces its association to plakoglobin. The binding sites of Tcf-4 for these two proteins were compared; whereas beta-catenin requires the N-terminal first 50 amino acids, plakoglobin interacts mainly with residues 51-80. Tcf-4-(51-80) binds plakoglobin in the region of armadillo repeats 1-6. Ternary complexes composed by beta-catenin/Tcf-4/plakoglobin could be detected in vitro, demonstrating that simultaneous binding of the two armadillo proteins to Tcf-4 is possible. Experiments performed using a Tcf-4 mutant with decreased interaction to plakoglobin demonstrated that binding to this protein negatively affected the transcriptional activity of Tcf-4. These results indicate that Tcf-4 contains two different sites for binding of beta-catenin and plakoglobin, and the interaction of the latter hinders the transcriptional activity of the complex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Base Sequence
  • Binding Sites
  • Casein Kinase II
  • Cytoskeletal Proteins / metabolism*
  • DNA Primers
  • Desmoplakins
  • Humans
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism
  • Trans-Activators*
  • Transcription Factors / metabolism*
  • beta Catenin
  • gamma Catenin

Substances

  • CTNNB1 protein, human
  • Cytoskeletal Proteins
  • DNA Primers
  • Desmoplakins
  • Trans-Activators
  • Transcription Factors
  • beta Catenin
  • gamma Catenin
  • Casein Kinase II
  • Protein Serine-Threonine Kinases