Anoplin, a novel antimicrobial peptide from the venom of the solitary wasp Anoplius samariensis

Biochim Biophys Acta. 2001 Nov 26;1550(1):70-80. doi: 10.1016/s0167-4838(01)00271-0.

Abstract

A novel antimicrobial peptide, anoplin, was purified from the venom of the solitary wasp Anoplius samariensis. The sequence was mostly analyzed by mass spectrometry, which was corroborated by solid-phase synthesis. Anoplin, composed of 10 amino acid residues, Gly-Leu-Leu-Lys-Arg-Ile-Lys-Thr-Leu-Leu-NH2, has a high homology to crabrolin and mastoparan-X, the mast cell degranulating peptides from social wasp venoms, and, therefore, can be predicted to adopt an amphipathic alpha-helix secondary structure. In fact, the circular dichroism (CD) spectra of anoplin in the presence of trifluoroethanol or sodium dodecyl sulfate showed a high content, up to 55%, of the alpha-helical conformation. A modeling study of anoplin based on its homology to mastoparan-X supported the CD results. Biological evaluation using the synthetic peptide revealed that this peptide exhibited potent activity in stimulating degranulation from rat peritoneal mast cells and broad-spectrum antimicrobial activity against both Gram-positive and Gram-negative bacteria. Therefore, this is the first antimicrobial component to be found in the solitary wasp venom and it may play a key role in preventing potential infection by microorganisms during prey consumption by their larvae. Moreover, this peptide is the smallest among the linear alpha-helical antimicrobial peptides hitherto found in nature, which is advantageous for chemical manipulation and medical application.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / isolation & purification*
  • Anti-Bacterial Agents / pharmacology
  • Antimicrobial Cationic Peptides
  • Cell Degranulation
  • Chromatography, High Pressure Liquid
  • Circular Dichroism
  • Female
  • Mast Cells / drug effects
  • Mast Cells / physiology
  • Microbial Sensitivity Tests
  • Models, Molecular
  • Oligopeptides / chemistry*
  • Oligopeptides / isolation & purification*
  • Oligopeptides / pharmacology
  • Rats
  • Sequence Alignment
  • Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
  • Wasp Venoms / chemistry*
  • Wasp Venoms / isolation & purification*
  • Wasp Venoms / pharmacology
  • Wasps

Substances

  • Anti-Bacterial Agents
  • Antimicrobial Cationic Peptides
  • Oligopeptides
  • Wasp Venoms
  • anoplin