Three-dimensional structure of the synaptotagmin 1 C2B-domain: synaptotagmin 1 as a phospholipid binding machine

Neuron. 2001 Dec 20;32(6):1057-69. doi: 10.1016/s0896-6273(01)00548-7.

Abstract

Synaptotagmin 1 probably functions as a Ca2+ sensor in neurotransmitter release via its two C2-domains, but no common Ca2+-dependent activity that could underlie a cooperative action between them has been described. The NMR structure of the C2B-domain now reveals a beta sandwich that exhibits striking similarities and differences with the C2A-domain. Whereas the bottom face of the C2B-domain has two additional alpha helices that may be involved in specialized Ca2+-independent functions, the top face binds two Ca2+ ions and is remarkably similar to the C2A-domain. Consistent with these results, but in contrast to previous studies, we find that the C2B-domain binds phospholipids in a Ca2+-dependent manner similarly to the C2A-domain. These results suggest a novel view of synaptotagmin function whereby the two C2-domains cooperate in a common activity, Ca2+-dependent phospholipid binding, to trigger neurotransmitter release.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites / physiology
  • Calcium / metabolism
  • Calcium-Binding Proteins*
  • Magnetic Resonance Spectroscopy
  • Membrane Glycoproteins / chemistry*
  • Membrane Glycoproteins / metabolism*
  • Molecular Sequence Data
  • Nerve Tissue Proteins / chemistry*
  • Nerve Tissue Proteins / metabolism*
  • Neurotransmitter Agents / metabolism
  • Phospholipids / metabolism*
  • Protein Structure, Tertiary
  • Structure-Activity Relationship
  • Synaptic Transmission / physiology
  • Synaptotagmin I
  • Synaptotagmins

Substances

  • Calcium-Binding Proteins
  • Membrane Glycoproteins
  • Nerve Tissue Proteins
  • Neurotransmitter Agents
  • Phospholipids
  • Synaptotagmin I
  • Synaptotagmins
  • Calcium

Associated data

  • PDB/1K5W