Chronic hypoxia remodels voltage-gated Ca2+ entry in a human airway chemoreceptor cell line

Neurosci Lett. 2002 Jan 25;318(2):69-72. doi: 10.1016/s0304-3940(01)02479-x.

Abstract

Arterial and airway chemoreceptors respond to acute hypoxia by depolarizing, thereby activating voltage-gated Ca2+ channels and so permitting Ca2+ entry to trigger transmitter release. Following periods of prolonged hypoxia, these cells undergo a form of remodelling which involves altered expression of ion channels. Here, we use microspectrofluorimetric recordings of voltage-gated Ca2+ entry (activated by exposure of cells to 50 mM K+) to show that chronic hypoxia suppresses such Ca2+ entry in model airway chemoreceptor (H146) cells. Furthermore, Ca2+ entry via L-type channels is suppressed, whilst entry via N-type channels is greatly enhanced. The suppressed response, together with dramatic remodelling of routes available for voltage-gated Ca2+ entry, is likely to alter significantly the acute O2 sensing properties of these cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcium / metabolism*
  • Calcium Channel Blockers / pharmacology
  • Calcium Channels / drug effects
  • Calcium Channels / metabolism*
  • Calcium Signaling / drug effects
  • Calcium Signaling / physiology*
  • Chemoreceptor Cells / drug effects
  • Chemoreceptor Cells / metabolism*
  • Chronic Disease
  • Humans
  • Hypoxia / metabolism*
  • Hypoxia / physiopathology
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Potassium / pharmacology
  • Respiratory System / drug effects
  • Respiratory System / metabolism*
  • Tumor Cells, Cultured

Substances

  • Calcium Channel Blockers
  • Calcium Channels
  • Potassium
  • Calcium