Comparative cytotoxicity of low-osmolar nonionic and high-osmolar ionic contrast media to dog gallbladder epithelial cells

Gastrointest Endosc. 2002 Mar;55(3):382-6. doi: 10.1067/mge.2002.121595.

Abstract

Background: Most studies of the adverse effects of x-ray contrast media used in ERCP have focused on post-ERCP pancreatitis. However, the biliary epithelial cells are also exposed to contrast media during ERCP and acute cholangitis is also a serious complication of ERCP. The present study compared the cytotoxicity with gallbladder epithelial cells of ionic and nonionic contrast agents.

Methods: A high-osmolar ionic contrast agent (meglumine ioxithalamate) and a low-osmolar nonionic contrast agent (iopromide) were tested. Monolayer cell cultures of dog gallbladder epithelial cells were used. The cells were exposed to the 2 contrast agents with increasing iodine concentration and osmolality for 2 days. Cell number, S-phase fraction, aneuploidy, and supernatant LDH activities were measured each day.

Results: Cell growth was more severely inhibited by ioxithalamate than iopromide (p < 0.05) and strongly dependent on the osmolality of contrast agent. The cytostatic effect estimated by S-phase fraction was more pronounced for ioxithalamate. Chromosomal damage determined by aneuploidy was more frequently detected with ioxithalamate.

Conclusions: High-osmolar ionic contrast media are more cytotoxic than low-osmolar nonionic contrast media to gallbladder epithelial cells. Animal and clinical studies are needed to estimate the clinical implications of these findings.

Publication types

  • Comparative Study
  • Evaluation Study

MeSH terms

  • Aneuploidy
  • Animals
  • Cell Count
  • Cell Cycle / drug effects
  • Cholangiopancreatography, Endoscopic Retrograde / adverse effects
  • Cholangitis / chemically induced
  • Contrast Media / administration & dosage
  • Contrast Media / toxicity*
  • Dogs
  • Epithelial Cells / drug effects
  • Gallbladder / cytology
  • Iohexol / administration & dosage
  • Iohexol / analogs & derivatives*
  • Iohexol / toxicity*
  • Iothalamate Meglumine / administration & dosage
  • Iothalamate Meglumine / toxicity*
  • Pancreatitis / chemically induced

Substances

  • Contrast Media
  • Iohexol
  • meglumine ioxithalamate
  • iopromide
  • Iothalamate Meglumine