cAMP regulation of Cl(-) and HCO(-)(3) secretion across rat fetal distal lung epithelial cells

Am J Physiol Lung Cell Mol Physiol. 2002 Apr;282(4):L650-8. doi: 10.1152/ajplung.00370.2001.

Abstract

We isolated and cultured fetal distal lung epithelial (FDLE) cells from 17- to 19-day rat fetuses and assayed for anion secretion in Ussing chambers. With symmetrical Ringer solutions, basal short-circuit currents (I(sc)) and transepithelial resistances were 7.9 +/- 0.5 microA/cm(2) and 1,018 +/- 73 Omega.cm(2), respectively (means +/- SE; n = 12). Apical amiloride (10 microM) inhibited basal I(sc) by approximately 50%. Subsequent addition of forskolin (10 microM) increased I(sc) from 3.9 +/- 0.63 microA/cm(2) to 7.51 +/- 0.2 microA/cm(2) (n = 12). Basolateral bumetanide (100 microM) decreased forskolin-stimulated I(sc) from 7.51 +/- 0.2 microA/cm(2) to 5.62 +/- 0.53, whereas basolateral 4,4'-dinitrostilbene-2,2'-disulfonate (5 mM), an inhibitor of HCO secretion, blocked the remaining I(sc). Forskolin addition evoked currents of similar fractional magnitudes in symmetrical Cl(-)- or HCO(-)(3)-free solutions; however, no response was seen using HCO(-)(3)- and Cl(-)-free solutions. The forskolin-stimulated I(sc) was inhibited by glibenclamide but not apical DIDS. Glibenclamide also blocked forskolin-induced I(sc) across monolayers having nystatin-permeablized basolateral membranes. Immunolocalization studies were consistent with the expression of cystic fibrosis transmembrane conductance regulator (CFTR) protein in FDLE cells. In aggregate, these findings indicate the presence of cAMP-activated Cl(-) and HCO(-)(3) secretion across rat FDLE cells mediated via CFTR.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amiloride / pharmacology
  • Animals
  • Bicarbonates / metabolism*
  • Bumetanide / pharmacology
  • Cell Polarity / physiology
  • Cells, Cultured
  • Chlorides / metabolism*
  • Colforsin / pharmacology
  • Cyclic AMP / metabolism*
  • Cystic Fibrosis Transmembrane Conductance Regulator / analysis
  • Cystic Fibrosis Transmembrane Conductance Regulator / metabolism
  • Diuretics / pharmacology
  • Epithelial Cells / chemistry
  • Epithelial Cells / metabolism
  • Extravascular Lung Water / metabolism
  • Immunohistochemistry
  • Ionophores / pharmacology
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Nystatin / pharmacology
  • Pulmonary Alveoli / cytology
  • Pulmonary Alveoli / metabolism*
  • Rats
  • Respiratory Mucosa / cytology
  • Respiratory Mucosa / metabolism*
  • Stilbenes / pharmacology

Substances

  • Bicarbonates
  • Chlorides
  • Diuretics
  • Ionophores
  • Stilbenes
  • Bumetanide
  • Cystic Fibrosis Transmembrane Conductance Regulator
  • Nystatin
  • Colforsin
  • 4,4'-dinitro-2,2'-stilbenedisulfonic acid
  • Amiloride
  • Cyclic AMP