Oncogenic H-Ras enhances DNA repair through the Ras/phosphatidylinositol 3-kinase/Rac1 pathway in NIH3T3 cells. Evidence for association with reactive oxygen species

J Biol Chem. 2002 May 31;277(22):19358-66. doi: 10.1074/jbc.M200933200. Epub 2002 Mar 7.

Abstract

This study investigated the role of oncogenic H-Ras in DNA repair capacity in NIH3T3 cells. Expression of dominant-positive H-Ras (V12-H-Ras) enhanced the host cell reactivation of luciferase activity from UV-irradiated and cisplatin-treated plasmids and also increased the unscheduled DNA synthesis following cisplatin or UV treatment of cells. This observed enhancement of DNA repair capacity was inhibited by transient transfection with dominant-negative H-Ras (N17-H-Ras) or Rac1 (N17-Rac1) plasmids. Moreover, stable transfection of dominant-positive Rac1 (V12-Rac1) further enhanced DNA repair capacity. Because reactive oxygen species (ROS) are known to be a downstream effector of oncogenic Ras, we examined the role of ROS in DNA repair capacity. We found that ROS production by V12-H-Ras expression was mediated by the Ras/phosphatidylinositol 3-kinase (PI3K)/Rac1/NADPH oxidase-dependent pathway and that pretreatment of V12-H-Ras-transformed cells with an antioxidant (N-acetylcysteine) and an NADPH oxidase inhibitor (diphenyleneiodonium) decreased DNA repair capacity. Similarly, treatment with PI3K inhibitors (wortmannin and LY294002) inhibited the ability of oncogenic H-Ras to enhance DNA repair capacity. Furthermore, inhibition of the Ras/PI3K/Rac1/NADPH oxidase pathway resulted in increased sensitivity to cisplatin and UV in V12-H-Ras-expressing NIH3T3 cells. Taken together, these results provide evidence that oncogenic H-Ras activates DNA repair capacity through the Ras/PI3K/Rac1/NADPH oxidase-dependent pathway and that increased ROS production via this signaling pathway is required for enhancement of the DNA repair capacity induced by oncogenic H-Ras.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3 Cells
  • Acetylcysteine / pharmacology
  • Androstadienes / pharmacology
  • Animals
  • Blotting, Western
  • Cell Line
  • Cell Survival
  • Chromones / pharmacology
  • Cisplatin / pharmacology
  • DNA / biosynthesis
  • DNA Repair*
  • Enzyme Inhibitors / pharmacology
  • Genes, ras / genetics*
  • Luciferases / metabolism
  • Mice
  • Morpholines / pharmacology
  • Phosphatidylinositol 3-Kinases / metabolism*
  • Plasmids / metabolism
  • Reactive Oxygen Species*
  • Signal Transduction
  • Time Factors
  • Transfection
  • Ultraviolet Rays
  • Wortmannin
  • rac1 GTP-Binding Protein / metabolism*
  • ras Proteins / metabolism*

Substances

  • Androstadienes
  • Chromones
  • Enzyme Inhibitors
  • Morpholines
  • Reactive Oxygen Species
  • 2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one
  • DNA
  • Luciferases
  • Phosphatidylinositol 3-Kinases
  • rac1 GTP-Binding Protein
  • ras Proteins
  • Cisplatin
  • Acetylcysteine
  • Wortmannin