Effects of tibolone and continuous combined hormone replacement therapy on mammographic breast density

Am J Obstet Gynecol. 2002 Apr;186(4):717-22. doi: 10.1067/mob.2002.121896.

Abstract

Objective: Our purpose was to compare the effects of tibolone, continuous combined hormone replacement therapy, and placebo on mammographic breast density.

Study design: A prospective, randomized, double-blind placebo-controlled study was performed. A total of 166 postmenopausal women were equally randomized to receive tibolone 2.5 mg, estradiol 2 mg/norethisterone acetate 1 mg (E(2)/NETA), or placebo. Mammograms were performed at baseline and after 6 months of treatment. Mammographic density was quantified according to the Wolfe classification and by the percentage area of the breast that had a dense pattern.

Results: An increase in mammographic density was much more common among women receiving continuous combined hormone replacement therapy (46%-50%) than among those receiving tibolone (2%-6%) and placebo (0%) treatment. The difference between E(2)/NETA and placebo was highly significant (P <.001). Treatment with tibolone did not differ from that with placebo. The relative risk of an increase in breast density for E(2)/NETA versus tibolone was found to be 8.3 (95% CI 2.7-25.0).

Conclusion: An increase in mammographic density should be regarded as an unwanted side effect of hormone replacement therapy. In contrast to estrogen/progestogen treatment, tibolone seems to exert little stimulation of breast tissue.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biopsy, Needle
  • Breast / pathology*
  • Double-Blind Method
  • Estradiol / administration & dosage
  • Estradiol / adverse effects
  • Estrogen Receptor Modulators / adverse effects*
  • Estrogen Receptor Modulators / therapeutic use
  • Estrogen Replacement Therapy / adverse effects*
  • Humans
  • Mammography*
  • Norethindrone / administration & dosage
  • Norethindrone / adverse effects
  • Norethindrone / analogs & derivatives*
  • Norethindrone Acetate
  • Norpregnenes / adverse effects*
  • Norpregnenes / therapeutic use
  • Placebos
  • Postmenopause*
  • Prospective Studies

Substances

  • Estrogen Receptor Modulators
  • Norpregnenes
  • Placebos
  • Estradiol
  • Norethindrone Acetate
  • tibolone
  • Norethindrone